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2Y0J

Triazoloquinazolines as a novel class of phosphodiesterase 10A (PDE10A) inhibitors, part 2, Lead-optimisation.

Resources
File formatFile name (file size)
PDBx/mmCIF2y0j.cif.gz Display(143.48 KB)
2y0j.cif
PDBx/mmJSONall2y0j.json.gz Display (Tree)(94.46 KB)
2y0j.json
no-atom2y0j-noatom.json.gz Display (Header)(16.61 KB)
2y0j-noatom.json
add only2y0j-plus.json.gz Display(1.14 KB)
2y0j-plus.json
PDBMLall2y0j.xml.gz Display(193.10 KB)
2y0j.xml
no-atom2y0j-noatom.xml.gz Display(36.48 KB)
2y0j-noatom.xml
ext-atom2y0j-extatom.xml.gz Display(118.75 KB)
2y0j-extatom.xml
pdb_nextgenallpdb_00002y0j_xyz-enrich.cif.gz Display(158.73 KB)
pdb_00002y0j_xyz-enrich.cif
no-atompdb_00002y0j_xyz-no-atom-enrich.xml.gz Display(50.96 KB)
pdb_00002y0j_xyz-no-atom-enrich.xml
ng-only2y0j-plus.json.gz Display(3.40 KB)
2y0j-plus.json
PDBpdb2y0j.ent.gz Display(111.70 KB)
pdb2y0j.ent
RDF2y0j.rdf.gz Visualize(104.66 KB)
2y0j.rdf
Structure factorsr2y0jsf.ent.gz Display(342.86 KB)
r2y0jsf.ent
Biological unit (mmCIF format)2y0j-assembly1.cif.gz Display(69.08 KB)
2y0j-assembly1.cif (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

2y0j-assembly2.cif.gz Display(69.35 KB)
2y0j-assembly2.cif (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)2y0j.pdb1.gz Display(54.05 KB)
2y0j.pdb1 (A)

*author and software defined assembly, 1 molecule(s) (monomeric)

2y0j.pdb2.gz Display(54.35 KB)
2y0j.pdb2 (B)

*author and software defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF2y0j_validation.pdf.gz Display(1.19 MB)
2y0j_validation.pdf
PDF-full2y0j_full_validation.pdf.gz Display(1.19 MB)
2y0j_full_validation.pdf
mmCIF2y0j_validation.cif.gz Display(41.16 KB)
2y0j_validation.cif
XML2y0j_validation.xml.gz Display(30.47 KB)
2y0j_validation.xml
PNG2y0j_multipercentile_validation.png.gz Display(168.25 KB)
2y0j_multipercentile_validation.png
SVG2y0j_multipercentile_validation.svg.gz Display(948.00 B)
2y0j_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)2y0j_validation_2fo-fc_map_coef.cif.gz Display(366.59 KB)
2y0j_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)2y0j_validation_fo-fc_map_coef.cif.gz Display(365.84 KB)
2y0j_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)2y0j_validation_2fo-fc_map_coef.mtz Visualize(594.92 KB)
fo-fc (MTZ)2y0j_validation_fo-fc_map_coef.mtz Visualize(594.92 KB)

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PDB entries from 2026-06-03

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