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1EAT

NONPEPTIDIC INHIBITORS OF HUMAN LEUKOCYTE ELASTASE. 5. DESIGN, SYNTHESIS, AND X-RAY CRYSTALLOGRAPHY OF A SERIES OF ORALLY ACTIVE 5-AMINO-PYRIMIDIN-6-ONE-CONTAINING TRIFLUOROMETHYLKETONES

Resources
File formatFile name (file size)
PDBx/mmCIF1eat.cif.gz Display(65.00 KB)
1eat.cif
PDBx/mmJSONall1eat.json.gz Display (Tree)(45.82 KB)
1eat.json
no-atom1eat-noatom.json.gz Display (Header)(14.03 KB)
1eat-noatom.json
add only1eat-plus.json.gz Display(1.72 KB)
1eat-plus.json
PDBMLall1eat.xml.gz Display(86.89 KB)
1eat.xml
no-atom1eat-noatom.xml.gz Display(25.84 KB)
1eat-noatom.xml
ext-atom1eat-extatom.xml.gz Display(45.14 KB)
1eat-extatom.xml
pdb_nextgenallpdb_00001eat_xyz-enrich.cif.gz Display(72.65 KB)
pdb_00001eat_xyz-enrich.cif
no-atompdb_00001eat_xyz-no-atom-enrich.xml.gz Display(35.31 KB)
pdb_00001eat_xyz-no-atom-enrich.xml
ng-only1eat-plus.json.gz Display(2.17 KB)
1eat-plus.json
PDBpdb1eat.ent.gz Display(46.11 KB)
pdb1eat.ent
RDF1eat.rdf.gz Visualize(74.98 KB)
1eat.rdf
Structure factorsr1eatsf.ent.gz Display(111.44 KB)
r1eatsf.ent
Biological unit (mmCIF format)1eat-assembly1.cif.gz Display(54.87 KB)
1eat-assembly1.cif (A)

*author defined assembly, 1 molecule(s) (monomeric)

Biological unit (PDB format)1eat.pdb1.gz Display(42.13 KB)
1eat.pdb1 (A)

*author defined assembly, 1 molecule(s) (monomeric)

Validation reportsPDF1eat_validation.pdf.gz Display(762.41 KB)
1eat_validation.pdf
PDF-full1eat_full_validation.pdf.gz Display(764.74 KB)
1eat_full_validation.pdf
mmCIF1eat_validation.cif.gz Display(17.37 KB)
1eat_validation.cif
XML1eat_validation.xml.gz Display(12.54 KB)
1eat_validation.xml
PNG1eat_multipercentile_validation.png.gz Display(150.07 KB)
1eat_multipercentile_validation.png
SVG1eat_multipercentile_validation.svg.gz Display(903.00 B)
1eat_multipercentile_validation.svg
EDMap2fo-fc (PDBx/mmCIF)1eat_validation_2fo-fc_map_coef.cif.gz Display(214.02 KB)
1eat_validation_2fo-fc_map_coef.cif
fo-fc (PDBx/mmCIF)1eat_validation_fo-fc_map_coef.cif.gz Display(193.41 KB)
1eat_validation_fo-fc_map_coef.cif
2fo-fc (MTZ)1eat_validation_2fo-fc_map_coef.mtz Visualize(369.24 KB)
fo-fc (MTZ)1eat_validation_fo-fc_map_coef.mtz Visualize(369.24 KB)

246704

PDB entries from 2025-12-24

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