Summary
| Title: | N-TERMINAL BROMODOMAIN OF HUMAN BRD2 WITH 3,5 dimethyl-4-phenyl-1,2- oxazole |
| Citation: | Bamborough, P.,Diallo, H.,Goodacre, J.D.,Gordon, L.,Lewis, A.,Seal, J.T.,Wilson, D.M.,Woodrow, M.D.,Chung, C.W. Fragment-Based Discovery of Bromodomain Inhibitors Part 2: Optimization of Phenylisoxazole Sulfonamides. J.Med.Chem., 55:587-, 2012 PubMed: 22136469DOI: 10.1021/JM201283Q |
| Experimental method: | X-RAY DIFFRACTION (1.78 Å) |
| Deposition date: | 2011-11-26 |
| Release date: | 2012-02-08 |
| Obsoletion date: | 2012-04-11 |
Timeline
Downloads
| File format | File name (file size) | ||
| PDBx/mmCIF | 4a9p.cif.gz Display(159.18 KB) 4a9p.cif | ||
| PDBx/mmJSON | no-atom | 4a9p-noatom.json.gz Display (Header)(10.35 KB) 4a9p-noatom.json | |
| PDBML | all | 4a9p.xml.gz Display(220.44 KB) 4a9p.xml | |
| PDB | pdb4a9p.ent.gz Display(133.43 KB) pdb4a9p.ent | ||
| Structure factors | r4a9psf.ent.gz Display(291.33 KB) r4a9psf.ent | ||






