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9FEH

Crystal structure of SARS-CoV-2 nsp14 methyltransferase domain in complex with the STM957 inhibitor

This is a non-PDB format compatible entry.
Functional Information from GO Data
ChainGOidnamespacecontents
A0004482molecular_functionmRNA 5'-cap (guanine-N7-)-methyltransferase activity
A0004532molecular_functionRNA exonuclease activity
A0008168molecular_functionmethyltransferase activity
A0043565molecular_functionsequence-specific DNA binding
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBinding site: {"evidences":[{"source":"PROSITE-ProRule","id":"PRU01299","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues4
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"36546776","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues1
DetailsSite: {"description":"Breakpoint for translocation to form ETV6-MDS2 in MDS"}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues1
DetailsSite: {"description":"Breakpoint for translocation to form PAX5-ETV6"}
ChainResidueDetails

239803

PDB entries from 2025-08-06

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