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9EHS

Structure of a human adenosine A3 receptor complex bound to the covalent antagonist LUF7602

This is a non-PDB format compatible entry.
Functional Information from PROSITE/UniProt
site_idPS00290
Number of Residues7
DetailsIG_MHC Immunoglobulins and major histocompatibility complex proteins signature. YICNVNH
ChainResidueDetails
HTYR208-HIS214
LTYR194-HIS200

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues23
DetailsTransmembrane: {"description":"Helical; Name=1","evidences":[{"source":"PubMed","id":"38627384","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"40825947","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"8X16","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"8X17","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBI","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EHS","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues26
DetailsTopological domain: {"description":"Cytoplasmic","evidences":[{"source":"PubMed","id":"38627384","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"40825947","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"8X16","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"8X17","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBI","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EHS","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues22
DetailsTransmembrane: {"description":"Helical; Name=2","evidences":[{"source":"PubMed","id":"38627384","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"40825947","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"8X16","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"8X17","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBI","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EHS","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues41
DetailsTopological domain: {"description":"Extracellular","evidences":[{"source":"PubMed","id":"38627384","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"40825947","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"8X16","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"8X17","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBI","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EHS","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues22
DetailsTransmembrane: {"description":"Helical; Name=3","evidences":[{"source":"PubMed","id":"38627384","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"40825947","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"8X16","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"8X17","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBI","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EHS","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues22
DetailsTransmembrane: {"description":"Helical; Name=4","evidences":[{"source":"PubMed","id":"38627384","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"40825947","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"8X16","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"8X17","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBI","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EHS","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI7
Number of Residues25
DetailsTransmembrane: {"description":"Helical; Name=5","evidences":[{"source":"PubMed","id":"38627384","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"40825947","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"8X16","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"8X17","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBI","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EHS","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI8
Number of Residues25
DetailsTransmembrane: {"description":"Helical; Name=6","evidences":[{"source":"PubMed","id":"38627384","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"40825947","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"8X16","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"8X17","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBI","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EHS","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI9
Number of Residues21
DetailsTransmembrane: {"description":"Helical; Name=7","evidences":[{"source":"PubMed","id":"38627384","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"40825947","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"8X16","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"8X17","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBH","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EBI","evidenceCode":"ECO:0007744"},{"source":"PDB","id":"9EHS","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI10
Number of Residues1
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"40825947","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"9EBH","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI11
Number of Residues1
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"39511145","evidenceCode":"ECO:0000305"}]}
ChainResidueDetails

site_idSWS_FT_FI12
Number of Residues2
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"P35342","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI13
Number of Residues1
DetailsGlycosylation: {"description":"N-linked (GlcNAc...) asparagine","evidences":[{"evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

250359

PDB entries from 2026-03-11

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