9E30
Discovery of Potent, Highly Selective and Efficacious SMARCA2 Degraders - Compound 13
This is a non-PDB format compatible entry.
Functional Information from GO Data
Functional Information from PROSITE/UniProt
site_id | PS00633 |
Number of Residues | 58 |
Details | BROMODOMAIN_1 Bromodomain signature. SevFiqlpSrkelp..EYYelIrkpVdfkkIkerirnhk..Yrslgdlekdvml.LchNAqtF |
Chain | Residue | Details |
A | SER1406-PHE1463 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 3 |
Details | Binding site: {"evidences":[{"source":"PubMed","id":"39570797","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"9E30","evidenceCode":"ECO:0007744"}]} |
Chain | Residue | Details |
site_id | SWS_FT_FI2 |
Number of Residues | 3 |
Details | Binding site: {"evidences":[{"source":"PubMed","id":"39570797","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"9E31","evidenceCode":"ECO:0007744"}]} |
Chain | Residue | Details |
site_id | SWS_FT_FI3 |
Number of Residues | 1 |
Details | Modified residue: {"description":"Phosphoserine","evidences":[{"source":"PubMed","id":"23186163","evidenceCode":"ECO:0007744"},{"source":"PubMed","id":"24275569","evidenceCode":"ECO:0007744"}]} |
Chain | Residue | Details |