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9CR7

Structure of human SETD8 in complex with covalent inhibitor AM2928

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues242
DetailsDomain: {"description":"SET","evidences":[{"source":"PROSITE-ProRule","id":"PRU00190","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsBinding site: {}
ChainResidueDetails

248942

PDB entries from 2026-02-11

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