Loading
PDBj
MenuPDBj@FacebookPDBj@X(formerly Twitter)PDBj@BlueSkyPDBj@YouTubewwPDB FoundationwwPDBDonate
RCSB PDBPDBeBMRBAdv. SearchSearch help

9BS9

Local refinement of DRD2 bound to LSD in complex with a mini-GoA and scFv16 obtained by cryo-electron microscopy (cryoEM)

Functional Information from GO Data
ChainGOidnamespacecontents
R0000139cellular_componentGolgi membrane
R0001591molecular_functiondopamine neurotransmitter receptor activity, coupled via Gi/Go
R0001659biological_processtemperature homeostasis
R0001666biological_processresponse to hypoxia
R0001669cellular_componentacrosomal vesicle
R0001963biological_processsynaptic transmission, dopaminergic
R0001965molecular_functionG-protein alpha-subunit binding
R0001975biological_processresponse to amphetamine
R0001976biological_processnervous system process involved in regulation of systemic arterial blood pressure
R0002027biological_processregulation of heart rate
R0002028biological_processregulation of sodium ion transport
R0002031biological_processG protein-coupled receptor internalization
R0002052biological_processpositive regulation of neuroblast proliferation
R0002092biological_processpositive regulation of receptor internalization
R0004930molecular_functionG protein-coupled receptor activity
R0004952molecular_functiondopamine neurotransmitter receptor activity
R0005102molecular_functionsignaling receptor binding
R0005515molecular_functionprotein binding
R0005886cellular_componentplasma membrane
R0005929cellular_componentcilium
R0006914biological_processautophagy
R0007165biological_processsignal transduction
R0007186biological_processG protein-coupled receptor signaling pathway
R0007188biological_processadenylate cyclase-modulating G protein-coupled receptor signaling pathway
R0007195biological_processadenylate cyclase-inhibiting dopamine receptor signaling pathway
R0007212biological_processG protein-coupled dopamine receptor signaling pathway
R0007270biological_processneuron-neuron synaptic transmission
R0007409biological_processaxonogenesis
R0007416biological_processsynapse assembly
R0007608biological_processsensory perception of smell
R0007616biological_processlong-term memory
R0007626biological_processlocomotory behavior
R0007628biological_processadult walking behavior
R0008104biological_processintracellular protein localization
R0008285biological_processnegative regulation of cell population proliferation
R0008306biological_processassociative learning
R0008542biological_processvisual learning
R0009410biological_processresponse to xenobiotic stimulus
R0009416biological_processresponse to light stimulus
R0009636biological_processresponse to toxic substance
R0010039biological_processresponse to iron ion
R0014059biological_processregulation of dopamine secretion
R0014854biological_processresponse to inactivity
R0016020cellular_componentmembrane
R0016055biological_processWnt signaling pathway
R0016328cellular_componentlateral plasma membrane
R0021756biological_processstriatum development
R0021769biological_processorbitofrontal cortex development
R0021853biological_processcerebral cortex GABAergic interneuron migration
R0021984biological_processadenohypophysis development
R0030139cellular_componentendocytic vesicle
R0030336biological_processnegative regulation of cell migration
R0030424cellular_componentaxon
R0030425cellular_componentdendrite
R0030432biological_processperistalsis
R0030672cellular_componentsynaptic vesicle membrane
R0030900biological_processforebrain development
R0031223biological_processauditory behavior
R0032228biological_processregulation of synaptic transmission, GABAergic
R0032355biological_processresponse to estradiol
R0032467biological_processpositive regulation of cytokinesis
R0032795molecular_functionheterotrimeric G-protein binding
R0032922biological_processcircadian regulation of gene expression
R0033602biological_processnegative regulation of dopamine secretion
R0034776biological_processresponse to histamine
R0035094biological_processresponse to nicotine
R0035240molecular_functiondopamine binding
R0035255molecular_functionionotropic glutamate receptor binding
R0035305biological_processnegative regulation of dephosphorylation
R0036126cellular_componentsperm flagellum
R0042220biological_processresponse to cocaine
R0042321biological_processnegative regulation of circadian sleep/wake cycle, sleep
R0042417biological_processdopamine metabolic process
R0042734cellular_componentpresynaptic membrane
R0042756biological_processdrinking behavior
R0042802molecular_functionidentical protein binding
R0043197cellular_componentdendritic spine
R0043204cellular_componentperikaryon
R0043266biological_processregulation of potassium ion transport
R0043278biological_processresponse to morphine
R0043408biological_processregulation of MAPK cascade
R0043679cellular_componentaxon terminus
R0044877molecular_functionprotein-containing complex binding
R0045211cellular_componentpostsynaptic membrane
R0045471biological_processresponse to ethanol
R0045745biological_processpositive regulation of G protein-coupled receptor signaling pathway
R0045776biological_processnegative regulation of blood pressure
R0045824biological_processnegative regulation of innate immune response
R0045944biological_processpositive regulation of transcription by RNA polymerase II
R0046676biological_processnegative regulation of insulin secretion
R0046717biological_processacid secretion
R0048148biological_processbehavioral response to cocaine
R0048149biological_processbehavioral response to ethanol
R0048169biological_processregulation of long-term neuronal synaptic plasticity
R0048678biological_processresponse to axon injury
R0048755biological_processbranching morphogenesis of a nerve
R0050482biological_processarachidonate secretion
R0050709biological_processnegative regulation of protein secretion
R0050769biological_processpositive regulation of neurogenesis
R0050805biological_processnegative regulation of synaptic transmission
R0051209biological_processrelease of sequestered calcium ion into cytosol
R0051240biological_processpositive regulation of multicellular organismal process
R0051481biological_processnegative regulation of cytosolic calcium ion concentration
R0051580biological_processregulation of neurotransmitter uptake
R0051584biological_processregulation of dopamine uptake involved in synaptic transmission
R0051586biological_processpositive regulation of dopamine uptake involved in synaptic transmission
R0051823biological_processregulation of synapse structural plasticity
R0051898biological_processnegative regulation of phosphatidylinositol 3-kinase/protein kinase B signal transduction
R0051952biological_processregulation of amine transport
R0051967biological_processnegative regulation of synaptic transmission, glutamatergic
R0060079biological_processexcitatory postsynaptic potential
R0060124biological_processpositive regulation of growth hormone secretion
R0060134biological_processprepulse inhibition
R0060158biological_processphospholipase C-activating dopamine receptor signaling pathway
R0060160biological_processnegative regulation of dopamine receptor signaling pathway
R0060170cellular_componentciliary membrane
R0070374biological_processpositive regulation of ERK1 and ERK2 cascade
R0071300biological_processcellular response to retinoic acid
R0071361biological_processcellular response to ethanol
R0090325biological_processregulation of locomotion involved in locomotory behavior
R0097305biological_processresponse to alcohol
R0097648cellular_componentG protein-coupled receptor complex
R0097730cellular_componentnon-motile cilium
R0098691cellular_componentdopaminergic synapse
R0098978cellular_componentglutamatergic synapse
R0098982cellular_componentGABA-ergic synapse
R0099170biological_processpostsynaptic modulation of chemical synaptic transmission
R0099171biological_processpresynaptic modulation of chemical synaptic transmission
R0160213biological_processbeta-arrestin-dependent dopamine receptor signaling pathway
R1900038biological_processnegative regulation of cellular response to hypoxia
R1900168biological_processpositive regulation of glial cell-derived neurotrophic factor production
R1900273biological_processpositive regulation of long-term synaptic potentiation
R1903530biological_processregulation of secretion by cell
R1990384biological_processhyaloid vascular plexus regression
Functional Information from PROSITE/UniProt
site_idPS00237
Number of Residues17
DetailsG_PROTEIN_RECEP_F1_1 G-protein coupled receptors family 1 signature. ASIlNLCAISIDRYTaV
ChainResidueDetails
RALA120-VAL136

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues22
DetailsTransmembrane: {"description":"Helical; Name=1","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues29
DetailsTopological domain: {"description":"Cytoplasmic","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues22
DetailsTransmembrane: {"description":"Helical; Name=2","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues29
DetailsTopological domain: {"description":"Extracellular","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues21
DetailsTransmembrane: {"description":"Helical; Name=3","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues20
DetailsTransmembrane: {"description":"Helical; Name=4","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI7
Number of Residues24
DetailsTransmembrane: {"description":"Helical; Name=5","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI8
Number of Residues21
DetailsTransmembrane: {"description":"Helical; Name=6","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI9
Number of Residues21
DetailsTransmembrane: {"description":"Helical; Name=7","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI10
Number of Residues2
DetailsSite: {"description":"Important for receptor activation","evidences":[{"evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

246905

PDB entries from 2025-12-31

PDB statisticsPDBj update infoContact PDBjnumon