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8XGA

Crystal structure of human Golgi resident glutaminyl cyclase in complex with (Z)-3-((1H-benzo[d]imidazol-5-yl)methylene)-4-((tetrahydro-2H-pyran-4-yl)oxy)indolin-2-one

This is a non-PDB format compatible entry.
Functional Information from GO Data
ChainGOidnamespacecontents
A0016603molecular_functionglutaminyl-peptide cyclotransferase activity
B0016603molecular_functionglutaminyl-peptide cyclotransferase activity
C0016603molecular_functionglutaminyl-peptide cyclotransferase activity
D0016603molecular_functionglutaminyl-peptide cyclotransferase activity
E0016603molecular_functionglutaminyl-peptide cyclotransferase activity
F0016603molecular_functionglutaminyl-peptide cyclotransferase activity
G0016603molecular_functionglutaminyl-peptide cyclotransferase activity
H0016603molecular_functionglutaminyl-peptide cyclotransferase activity
I0016603molecular_functionglutaminyl-peptide cyclotransferase activity
J0016603molecular_functionglutaminyl-peptide cyclotransferase activity
K0016603molecular_functionglutaminyl-peptide cyclotransferase activity
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues22
DetailsActive site: {"description":"Proton acceptor","evidences":[{"source":"UniProtKB","id":"Q16769","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues33
DetailsBinding site: {"evidences":[{"source":"UniProtKB","id":"Q16769","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

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PDB entries from 2025-11-05

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