8W7E
Design, synthesis and biological evaluations of novel small molecular hyper-activators of human caseinolytic peptidase P (hClpP)
Functional Information from PROSITE/UniProt
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 14 |
Details | ACT_SITE: Nucleophile => ECO:0000269|PubMed:11923310 |
Chain | Residue | Details |
A | SER153 | |
J | SER153 | |
K | SER153 | |
L | SER153 | |
M | SER153 | |
N | SER153 | |
B | SER153 | |
C | SER153 | |
D | SER153 | |
E | SER153 | |
F | SER153 | |
G | SER153 | |
H | SER153 | |
I | SER153 |
site_id | SWS_FT_FI2 |
Number of Residues | 14 |
Details | ACT_SITE: ACT_SITE => ECO:0000250 |
Chain | Residue | Details |
A | HIS178 | |
J | HIS178 | |
K | HIS178 | |
L | HIS178 | |
M | HIS178 | |
N | HIS178 | |
B | HIS178 | |
C | HIS178 | |
D | HIS178 | |
E | HIS178 | |
F | HIS178 | |
G | HIS178 | |
H | HIS178 | |
I | HIS178 |
site_id | SWS_FT_FI3 |
Number of Residues | 14 |
Details | MOD_RES: N6-succinyllysine => ECO:0000250|UniProtKB:O88696 |
Chain | Residue | Details |
A | LYS200 | |
J | LYS200 | |
K | LYS200 | |
L | LYS200 | |
M | LYS200 | |
N | LYS200 | |
B | LYS200 | |
C | LYS200 | |
D | LYS200 | |
E | LYS200 | |
F | LYS200 | |
G | LYS200 | |
H | LYS200 | |
I | LYS200 |
site_id | SWS_FT_FI4 |
Number of Residues | 14 |
Details | MOD_RES: N6-acetyllysine => ECO:0007744|PubMed:19608861 |
Chain | Residue | Details |
A | LYS211 | |
J | LYS211 | |
K | LYS211 | |
L | LYS211 | |
M | LYS211 | |
N | LYS211 | |
B | LYS211 | |
C | LYS211 | |
D | LYS211 | |
E | LYS211 | |
F | LYS211 | |
G | LYS211 | |
H | LYS211 | |
I | LYS211 |