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8TQP

HIV-CA Disulfide linked Hexamer bound to Quinazolin-4-one Scaffold inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0016032biological_processviral process
B0016032biological_processviral process
C0016032biological_processviral process
D0016032biological_processviral process
E0016032biological_processviral process
F0016032biological_processviral process
G0016032biological_processviral process
H0016032biological_processviral process
I0016032biological_processviral process
J0016032biological_processviral process
K0016032biological_processviral process
L0016032biological_processviral process
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues12
DetailsSITE: Cis/trans isomerization of proline peptide bond; by human PPIA/CYPA => ECO:0000250
ChainResidueDetails
AGLY89
KGLY89
LGLY89
HGLY89
BGLY89
CGLY89
DGLY89
EGLY89
FGLY89
GGLY89
IGLY89
JGLY89

site_idSWS_FT_FI2
Number of Residues12
DetailsSITE: Cleavage; by viral protease => ECO:0000250
ChainResidueDetails
ALEU231
KLEU231
LLEU231
HLEU231
BLEU231
CLEU231
DLEU231
ELEU231
FLEU231
GLEU231
ILEU231
JLEU231

site_idSWS_FT_FI3
Number of Residues12
DetailsMOD_RES: Phosphoserine; by host MAPK1 => ECO:0000269|PubMed:24509437
ChainResidueDetails
ASER16
KSER16
LSER16
HSER16
BSER16
CSER16
DSER16
ESER16
FSER16
GSER16
ISER16
JSER16

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PDB entries from 2024-07-17

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