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8IHK

Cryo-EM structure of HCA3-Gi complex with acifran (local)

Functional Information from GO Data
ChainGOidnamespacecontents
R0004930molecular_functionG protein-coupled receptor activity
R0005506molecular_functioniron ion binding
R0005886cellular_componentplasma membrane
R0007186biological_processG protein-coupled receptor signaling pathway
R0009055molecular_functionelectron transfer activity
R0016020cellular_componentmembrane
R0020037molecular_functionheme binding
R0022900biological_processelectron transport chain
R0030054cellular_componentcell junction
R0042597cellular_componentperiplasmic space
R0046872molecular_functionmetal ion binding
R0070553molecular_functionnicotinic acid receptor activity
Functional Information from PROSITE/UniProt
site_idPS00237
Number of Residues17
DetailsG_PROTEIN_RECEP_F1_1 G-protein coupled receptors family 1 signature. GSIiFLTVVAVDRYFrV
ChainResidueDetails
RGLY113-VAL129

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsBINDING: axial binding residue
ChainResidueDetails
RTRP-98
RILE-3

site_idSWS_FT_FI2
Number of Residues21
DetailsTRANSMEM: Helical; Name=1 => ECO:0000255
ChainResidueDetails
RVAL29-TRP50

site_idSWS_FT_FI3
Number of Residues144
DetailsTOPO_DOM: Cytoplasmic => ECO:0000255
ChainResidueDetails
RILE51-ARG63
RASP124-TRP142
RARG210-VAL236
RPRO299-GLU387

site_idSWS_FT_FI4
Number of Residues21
DetailsTRANSMEM: Helical; Name=2 => ECO:0000255
ChainResidueDetails
RILE64-ASP85

site_idSWS_FT_FI5
Number of Residues62
DetailsTOPO_DOM: Extracellular => ECO:0000255
ChainResidueDetails
RTYR86-LEU102
RLYS164-LEU194
RLEU257-ASP273

site_idSWS_FT_FI6
Number of Residues20
DetailsTRANSMEM: Helical; Name=3 => ECO:0000255
ChainResidueDetails
RVAL103-VAL123

site_idSWS_FT_FI7
Number of Residues20
DetailsTRANSMEM: Helical; Name=4 => ECO:0000255
ChainResidueDetails
RTHR143-LEU163

site_idSWS_FT_FI8
Number of Residues14
DetailsTRANSMEM: Helical; Name=5 => ECO:0000255
ChainResidueDetails
RLEU195-ALA209

site_idSWS_FT_FI9
Number of Residues19
DetailsTRANSMEM: Helical; Name=6 => ECO:0000255
ChainResidueDetails
RALA237-TRP256

site_idSWS_FT_FI10
Number of Residues24
DetailsTRANSMEM: Helical; Name=7 => ECO:0000255
ChainResidueDetails
RLEU274-SER298

223166

PDB entries from 2024-07-31

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