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8DKS

IRAK4 IN COMPLEX WITH COMPOUND #3

Functional Information from GO Data
ChainGOidnamespacecontents
A0000166molecular_functionnucleotide binding
A0000287molecular_functionmagnesium ion binding
A0002224biological_processtoll-like receptor signaling pathway
A0002376biological_processimmune system process
A0002446biological_processneutrophil mediated immunity
A0002755biological_processMyD88-dependent toll-like receptor signaling pathway
A0004672molecular_functionprotein kinase activity
A0004674molecular_functionprotein serine/threonine kinase activity
A0005149molecular_functioninterleukin-1 receptor binding
A0005515molecular_functionprotein binding
A0005524molecular_functionATP binding
A0005615cellular_componentextracellular space
A0005634cellular_componentnucleus
A0005737cellular_componentcytoplasm
A0005829cellular_componentcytosol
A0005886cellular_componentplasma membrane
A0006468biological_processprotein phosphorylation
A0007165biological_processsignal transduction
A0007249biological_processcanonical NF-kappaB signal transduction
A0007254biological_processJNK cascade
A0008063biological_processToll signaling pathway
A0009986cellular_componentcell surface
A0010008cellular_componentendosome membrane
A0016301molecular_functionkinase activity
A0016740molecular_functiontransferase activity
A0019221biological_processcytokine-mediated signaling pathway
A0019897cellular_componentextrinsic component of plasma membrane
A0019901molecular_functionprotein kinase binding
A0031663biological_processlipopolysaccharide-mediated signaling pathway
A0034142biological_processtoll-like receptor 4 signaling pathway
A0034162biological_processtoll-like receptor 9 signaling pathway
A0035556biological_processintracellular signal transduction
A0038172biological_processinterleukin-33-mediated signaling pathway
A0043123biological_processpositive regulation of canonical NF-kappaB signal transduction
A0043405biological_processregulation of MAP kinase activity
A0044546biological_processNLRP3 inflammasome complex assembly
A0045087biological_processinnate immune response
A0048661biological_processpositive regulation of smooth muscle cell proliferation
A0070498biological_processinterleukin-1-mediated signaling pathway
A0106310molecular_functionprotein serine kinase activity
A1990266biological_processneutrophil migration
B0000166molecular_functionnucleotide binding
B0000287molecular_functionmagnesium ion binding
B0002224biological_processtoll-like receptor signaling pathway
B0002376biological_processimmune system process
B0002446biological_processneutrophil mediated immunity
B0002755biological_processMyD88-dependent toll-like receptor signaling pathway
B0004672molecular_functionprotein kinase activity
B0004674molecular_functionprotein serine/threonine kinase activity
B0005149molecular_functioninterleukin-1 receptor binding
B0005515molecular_functionprotein binding
B0005524molecular_functionATP binding
B0005615cellular_componentextracellular space
B0005634cellular_componentnucleus
B0005737cellular_componentcytoplasm
B0005829cellular_componentcytosol
B0005886cellular_componentplasma membrane
B0006468biological_processprotein phosphorylation
B0007165biological_processsignal transduction
B0007249biological_processcanonical NF-kappaB signal transduction
B0007254biological_processJNK cascade
B0008063biological_processToll signaling pathway
B0009986cellular_componentcell surface
B0010008cellular_componentendosome membrane
B0016301molecular_functionkinase activity
B0016740molecular_functiontransferase activity
B0019221biological_processcytokine-mediated signaling pathway
B0019897cellular_componentextrinsic component of plasma membrane
B0019901molecular_functionprotein kinase binding
B0031663biological_processlipopolysaccharide-mediated signaling pathway
B0034142biological_processtoll-like receptor 4 signaling pathway
B0034162biological_processtoll-like receptor 9 signaling pathway
B0035556biological_processintracellular signal transduction
B0038172biological_processinterleukin-33-mediated signaling pathway
B0043123biological_processpositive regulation of canonical NF-kappaB signal transduction
B0043405biological_processregulation of MAP kinase activity
B0044546biological_processNLRP3 inflammasome complex assembly
B0045087biological_processinnate immune response
B0048661biological_processpositive regulation of smooth muscle cell proliferation
B0070498biological_processinterleukin-1-mediated signaling pathway
B0106310molecular_functionprotein serine kinase activity
B1990266biological_processneutrophil migration
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsActive site: {"description":"Proton acceptor","evidences":[{"source":"PROSITE-ProRule","id":"PRU00159","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues16
DetailsBinding site: {"evidences":[{"source":"PROSITE-ProRule","id":"PRU00159","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues10
DetailsBinding site: {}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues2
DetailsModified residue: {"description":"Phosphoserine","evidences":[{"source":"PubMed","id":"17161373","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"17312103","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

246704

PDB entries from 2025-12-24

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