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8DKS

IRAK4 IN COMPLEX WITH COMPOUND #3

Functional Information from GO Data
ChainGOidnamespacecontents
A0000287molecular_functionmagnesium ion binding
A0002224biological_processtoll-like receptor signaling pathway
A0002446biological_processneutrophil mediated immunity
A0002755biological_processMyD88-dependent toll-like receptor signaling pathway
A0004672molecular_functionprotein kinase activity
A0004674molecular_functionprotein serine/threonine kinase activity
A0005149molecular_functioninterleukin-1 receptor binding
A0005515molecular_functionprotein binding
A0005524molecular_functionATP binding
A0005615cellular_componentextracellular space
A0005634cellular_componentnucleus
A0005737cellular_componentcytoplasm
A0005829cellular_componentcytosol
A0005886cellular_componentplasma membrane
A0006468biological_processprotein phosphorylation
A0006950biological_processresponse to stress
A0007165biological_processsignal transduction
A0007166biological_processcell surface receptor signaling pathway
A0007254biological_processJNK cascade
A0008063biological_processToll signaling pathway
A0009986cellular_componentcell surface
A0010008cellular_componentendosome membrane
A0016301molecular_functionkinase activity
A0019221biological_processcytokine-mediated signaling pathway
A0019897cellular_componentextrinsic component of plasma membrane
A0019901molecular_functionprotein kinase binding
A0031349biological_processpositive regulation of defense response
A0034142biological_processtoll-like receptor 4 signaling pathway
A0034162biological_processtoll-like receptor 9 signaling pathway
A0035556biological_processintracellular signal transduction
A0038172biological_processinterleukin-33-mediated signaling pathway
A0043123biological_processpositive regulation of canonical NF-kappaB signal transduction
A0045087biological_processinnate immune response
A0048661biological_processpositive regulation of smooth muscle cell proliferation
A0070498biological_processinterleukin-1-mediated signaling pathway
A0071222biological_processcellular response to lipopolysaccharide
A0106310molecular_functionprotein serine kinase activity
A1990266biological_processneutrophil migration
B0000287molecular_functionmagnesium ion binding
B0002224biological_processtoll-like receptor signaling pathway
B0002446biological_processneutrophil mediated immunity
B0002755biological_processMyD88-dependent toll-like receptor signaling pathway
B0004672molecular_functionprotein kinase activity
B0004674molecular_functionprotein serine/threonine kinase activity
B0005149molecular_functioninterleukin-1 receptor binding
B0005515molecular_functionprotein binding
B0005524molecular_functionATP binding
B0005615cellular_componentextracellular space
B0005634cellular_componentnucleus
B0005737cellular_componentcytoplasm
B0005829cellular_componentcytosol
B0005886cellular_componentplasma membrane
B0006468biological_processprotein phosphorylation
B0006950biological_processresponse to stress
B0007165biological_processsignal transduction
B0007166biological_processcell surface receptor signaling pathway
B0007254biological_processJNK cascade
B0008063biological_processToll signaling pathway
B0009986cellular_componentcell surface
B0010008cellular_componentendosome membrane
B0016301molecular_functionkinase activity
B0019221biological_processcytokine-mediated signaling pathway
B0019897cellular_componentextrinsic component of plasma membrane
B0019901molecular_functionprotein kinase binding
B0031349biological_processpositive regulation of defense response
B0034142biological_processtoll-like receptor 4 signaling pathway
B0034162biological_processtoll-like receptor 9 signaling pathway
B0035556biological_processintracellular signal transduction
B0038172biological_processinterleukin-33-mediated signaling pathway
B0043123biological_processpositive regulation of canonical NF-kappaB signal transduction
B0045087biological_processinnate immune response
B0048661biological_processpositive regulation of smooth muscle cell proliferation
B0070498biological_processinterleukin-1-mediated signaling pathway
B0071222biological_processcellular response to lipopolysaccharide
B0106310molecular_functionprotein serine kinase activity
B1990266biological_processneutrophil migration
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE: Proton acceptor => ECO:0000255|PROSITE-ProRule:PRU00159
ChainResidueDetails
AASP311
BASP311

site_idSWS_FT_FI2
Number of Residues2
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00159
ChainResidueDetails
AMET192
BMET192

site_idSWS_FT_FI3
Number of Residues6
DetailsBINDING:
ChainResidueDetails
ALYS213
ALYS313
AASP329
BLYS213
BLYS313
BASP329

site_idSWS_FT_FI4
Number of Residues2
DetailsMOD_RES: N-acetylmethionine => ECO:0007744|PubMed:22814378
ChainResidueDetails
AMET1
BMET1

site_idSWS_FT_FI5
Number of Residues2
DetailsMOD_RES: N6-acetyllysine => ECO:0007744|PubMed:19608861
ChainResidueDetails
ALYS34
BLYS34

site_idSWS_FT_FI6
Number of Residues2
DetailsMOD_RES: Phosphothreonine => ECO:0000269|PubMed:17312103, ECO:0000269|Ref.32
ChainResidueDetails
ATHR342
BTHR342

site_idSWS_FT_FI7
Number of Residues2
DetailsMOD_RES: Phosphothreonine => ECO:0000269|PubMed:17161373, ECO:0000269|PubMed:17312103, ECO:0000269|Ref.32
ChainResidueDetails
ATHR345
BTHR345

site_idSWS_FT_FI8
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0000269|PubMed:17161373, ECO:0000269|PubMed:17312103
ChainResidueDetails
ASEP346
BSEP346

223532

PDB entries from 2024-08-07

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