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7XGE

Crystal structure of MCL-1 in complex with computationally designed inhibitor protein

Functional Information from GO Data
ChainGOidnamespacecontents
B0042981biological_processregulation of apoptotic process
D0042981biological_processregulation of apoptotic process
F0042981biological_processregulation of apoptotic process
H0042981biological_processregulation of apoptotic process
Functional Information from PROSITE/UniProt
site_idPS01080
Number of Residues20
DetailsBH1 Apoptosis regulator, Bcl-2 family BH1 motif signature. VFsDGvtNWGRIVTLIsFGA
ChainResidueDetails
BVAL85-ALA104

site_idPS01258
Number of Residues12
DetailsBH2 Apoptosis regulator, Bcl-2 family BH2 motif signature. WLvkqRGWDgFV
ChainResidueDetails
BTRP137-VAL148

site_idPS01259
Number of Residues15
DetailsBH3 Apoptosis regulator, Bcl-2 family BH3 motif signature. AletLRrVGDGVQRN
ChainResidueDetails
BALA41-ASN55

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues56
DetailsMotif: {"description":"BH3"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues80
DetailsMotif: {"description":"BH1"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues60
DetailsMotif: {"description":"BH2"}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues5
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in ubiquitin)"}
ChainResidueDetails

243911

PDB entries from 2025-10-29

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