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7W2F

An open-like conformation of the sigma-1 receptor from Xenopus laevis complexed with PRE084 by co-crystallization

Functional Information from GO Data
ChainGOidnamespacecontents
A0005634cellular_componentnucleus
A0005635cellular_componentnuclear envelope
A0005637cellular_componentnuclear inner membrane
A0005640cellular_componentnuclear outer membrane
A0005783cellular_componentendoplasmic reticulum
A0005789cellular_componentendoplasmic reticulum membrane
A0006696biological_processergosterol biosynthetic process
A0006869biological_processlipid transport
A0016020cellular_componentmembrane
A0031410cellular_componentcytoplasmic vesicle
B0005634cellular_componentnucleus
B0005635cellular_componentnuclear envelope
B0005637cellular_componentnuclear inner membrane
B0005640cellular_componentnuclear outer membrane
B0005783cellular_componentendoplasmic reticulum
B0005789cellular_componentendoplasmic reticulum membrane
B0006696biological_processergosterol biosynthetic process
B0006869biological_processlipid transport
B0016020cellular_componentmembrane
B0031410cellular_componentcytoplasmic vesicle
C0005634cellular_componentnucleus
C0005635cellular_componentnuclear envelope
C0005637cellular_componentnuclear inner membrane
C0005640cellular_componentnuclear outer membrane
C0005783cellular_componentendoplasmic reticulum
C0005789cellular_componentendoplasmic reticulum membrane
C0006696biological_processergosterol biosynthetic process
C0006869biological_processlipid transport
C0016020cellular_componentmembrane
C0031410cellular_componentcytoplasmic vesicle
D0005634cellular_componentnucleus
D0005635cellular_componentnuclear envelope
D0005637cellular_componentnuclear inner membrane
D0005640cellular_componentnuclear outer membrane
D0005783cellular_componentendoplasmic reticulum
D0005789cellular_componentendoplasmic reticulum membrane
D0006696biological_processergosterol biosynthetic process
D0006869biological_processlipid transport
D0016020cellular_componentmembrane
D0031410cellular_componentcytoplasmic vesicle
E0005634cellular_componentnucleus
E0005635cellular_componentnuclear envelope
E0005637cellular_componentnuclear inner membrane
E0005640cellular_componentnuclear outer membrane
E0005783cellular_componentendoplasmic reticulum
E0005789cellular_componentendoplasmic reticulum membrane
E0006696biological_processergosterol biosynthetic process
E0006869biological_processlipid transport
E0016020cellular_componentmembrane
E0031410cellular_componentcytoplasmic vesicle
F0005634cellular_componentnucleus
F0005635cellular_componentnuclear envelope
F0005637cellular_componentnuclear inner membrane
F0005640cellular_componentnuclear outer membrane
F0005783cellular_componentendoplasmic reticulum
F0005789cellular_componentendoplasmic reticulum membrane
F0006696biological_processergosterol biosynthetic process
F0006869biological_processlipid transport
F0016020cellular_componentmembrane
F0031410cellular_componentcytoplasmic vesicle
G0005634cellular_componentnucleus
G0005635cellular_componentnuclear envelope
G0005637cellular_componentnuclear inner membrane
G0005640cellular_componentnuclear outer membrane
G0005783cellular_componentendoplasmic reticulum
G0005789cellular_componentendoplasmic reticulum membrane
G0006696biological_processergosterol biosynthetic process
G0006869biological_processlipid transport
G0016020cellular_componentmembrane
G0031410cellular_componentcytoplasmic vesicle
H0005634cellular_componentnucleus
H0005635cellular_componentnuclear envelope
H0005637cellular_componentnuclear inner membrane
H0005640cellular_componentnuclear outer membrane
H0005783cellular_componentendoplasmic reticulum
H0005789cellular_componentendoplasmic reticulum membrane
H0006696biological_processergosterol biosynthetic process
H0006869biological_processlipid transport
H0016020cellular_componentmembrane
H0031410cellular_componentcytoplasmic vesicle
I0005634cellular_componentnucleus
I0005635cellular_componentnuclear envelope
I0005637cellular_componentnuclear inner membrane
I0005640cellular_componentnuclear outer membrane
I0005783cellular_componentendoplasmic reticulum
I0005789cellular_componentendoplasmic reticulum membrane
I0006696biological_processergosterol biosynthetic process
I0006869biological_processlipid transport
I0016020cellular_componentmembrane
I0031410cellular_componentcytoplasmic vesicle
J0005634cellular_componentnucleus
J0005635cellular_componentnuclear envelope
J0005637cellular_componentnuclear inner membrane
J0005640cellular_componentnuclear outer membrane
J0005783cellular_componentendoplasmic reticulum
J0005789cellular_componentendoplasmic reticulum membrane
J0006696biological_processergosterol biosynthetic process
J0006869biological_processlipid transport
J0016020cellular_componentmembrane
J0031410cellular_componentcytoplasmic vesicle
K0005634cellular_componentnucleus
K0005635cellular_componentnuclear envelope
K0005637cellular_componentnuclear inner membrane
K0005640cellular_componentnuclear outer membrane
K0005783cellular_componentendoplasmic reticulum
K0005789cellular_componentendoplasmic reticulum membrane
K0006696biological_processergosterol biosynthetic process
K0006869biological_processlipid transport
K0016020cellular_componentmembrane
K0031410cellular_componentcytoplasmic vesicle
L0005634cellular_componentnucleus
L0005635cellular_componentnuclear envelope
L0005637cellular_componentnuclear inner membrane
L0005640cellular_componentnuclear outer membrane
L0005783cellular_componentendoplasmic reticulum
L0005789cellular_componentendoplasmic reticulum membrane
L0006696biological_processergosterol biosynthetic process
L0006869biological_processlipid transport
L0016020cellular_componentmembrane
L0031410cellular_componentcytoplasmic vesicle
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues36
DetailsTOPO_DOM: Lumenal => ECO:0000250|UniProtKB:Q99720
ChainResidueDetails
AMET1-TRP4
JMET1-TRP4
KMET1-TRP4
LMET1-TRP4
BMET1-TRP4
CMET1-TRP4
DMET1-TRP4
EMET1-TRP4
FMET1-TRP4
GMET1-TRP4
HMET1-TRP4
IMET1-TRP4

site_idSWS_FT_FI2
Number of Residues264
DetailsTRANSMEM: Helical => ECO:0000250|UniProtKB:Q99720
ChainResidueDetails
ALEU5-LEU27
JLEU5-LEU27
KLEU5-LEU27
LLEU5-LEU27
BLEU5-LEU27
CLEU5-LEU27
DLEU5-LEU27
ELEU5-LEU27
FLEU5-LEU27
GLEU5-LEU27
HLEU5-LEU27
ILEU5-LEU27

site_idSWS_FT_FI3
Number of Residues2316
DetailsTOPO_DOM: Cytoplasmic => ECO:0000250|UniProtKB:Q99720
ChainResidueDetails
ASER28-PHE221
JSER28-PHE221
KSER28-PHE221
LSER28-PHE221
BSER28-PHE221
CSER28-PHE221
DSER28-PHE221
ESER28-PHE221
FSER28-PHE221
GSER28-PHE221
HSER28-PHE221
ISER28-PHE221

site_idSWS_FT_FI4
Number of Residues24
DetailsSITE: Important for ligand binding => ECO:0000250|UniProtKB:Q99720
ChainResidueDetails
AASP123
EGLU169
FASP123
FGLU169
GASP123
GGLU169
HASP123
HGLU169
IASP123
IGLU169
JASP123
AGLU169
JGLU169
KASP123
KGLU169
LASP123
LGLU169
BASP123
BGLU169
CASP123
CGLU169
DASP123
DGLU169
EASP123

219869

PDB entries from 2024-05-15

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