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7UUU

First bromodomain of BRDT liganded with compound 2c

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SwpFqrpvDavklqlpDYYtiIknpMdlntIkkrlenky..Yakaseciedfnt.MfsNCylY
ChainResidueDetails
ASER49-TYR108

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsBINDING: BINDING => ECO:0000269|PubMed:22901802, ECO:0007744|PDB:4FLP
ChainResidueDetails
AASN109

site_idSWS_FT_FI2
Number of Residues2
DetailsSITE: Histone H4K5ac binding => ECO:0000250|UniProtKB:Q91Y44
ChainResidueDetails
AASN109
AASP114

237992

PDB entries from 2025-06-25

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