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7URD

Human PORCN in complex with LGK974 and WNT3A peptide

Functional Information from GO Data
ChainGOidnamespacecontents
A0005783cellular_componentendoplasmic reticulum
A0005789cellular_componentendoplasmic reticulum membrane
A0006497biological_processprotein lipidation
A0009100biological_processglycoprotein metabolic process
A0016020cellular_componentmembrane
A0016055biological_processWnt signaling pathway
A0016746molecular_functionacyltransferase activity
A0017147molecular_functionWnt-protein binding
A0030258biological_processlipid modification
A0032281cellular_componentAMPA glutamate receptor complex
A0045234biological_processprotein palmitoleylation
A0061355biological_processWnt protein secretion
A0098978cellular_componentglutamatergic synapse
A0099072biological_processregulation of postsynaptic membrane neurotransmitter receptor levels
A1990698molecular_functionpalmitoleoyltransferase activity
B0005102molecular_functionsignaling receptor binding
B0005576cellular_componentextracellular region
B0007275biological_processmulticellular organism development
B0016055biological_processWnt signaling pathway
Functional Information from PROSITE/UniProt
site_idPS00246
Number of Residues10
DetailsWNT1 Wnt-1 family signature. CKCHGLSGsC
ChainResidueDetails
BCYS203-CYS212

site_idPS00290
Number of Residues7
DetailsIG_MHC Immunoglobulins and major histocompatibility complex proteins signature. YICNVNH
ChainResidueDetails
HTYR219-HIS225
LTYR212-HIS218

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsLIPID: O-palmitoleoyl serine; by PORCN => ECO:0000269|PubMed:20826466, ECO:0000269|PubMed:21244856, ECO:0000269|PubMed:24292069, ECO:0000269|PubMed:25731175
ChainResidueDetails
BSER209
APHE67-PHE87
AGLY96-ASP116
AVAL153-PHE173
ALEU199-ILE219
AVAL253-ASP273
APHE338-VAL358
APHE397-ASP417

site_idSWS_FT_FI2
Number of Residues131
DetailsTOPO_DOM: Extracellular => ECO:0000255
ChainResidueDetails
ACYS39-HIS66
ATHR117-PRO152
APRO220-PHE252
ALEU359-LEU396

site_idSWS_FT_FI3
Number of Residues94
DetailsTOPO_DOM: Cytoplasmic => ECO:0000255
ChainResidueDetails
ALEU88-ARG95
AHIS174-ALA198
AHIS274-GLY337

site_idSWS_FT_FI4
Number of Residues1
DetailsACT_SITE: ACT_SITE => ECO:0000269|PubMed:24292069
ChainResidueDetails
AHIS341

site_idSWS_FT_FI5
Number of Residues1
DetailsLIPID: S-palmitoyl cysteine => ECO:0000269|PubMed:24292069
ChainResidueDetails
ACYS187

222624

PDB entries from 2024-07-17

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