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7UKH

Human Kv4.2-KChIP2-DPP6 channel complex in an open state, intracellular region

Functional Information from GO Data
ChainGOidnamespacecontents
A0005216molecular_functionmonoatomic ion channel activity
A0005249molecular_functionvoltage-gated potassium channel activity
A0006811biological_processmonoatomic ion transport
A0006813biological_processpotassium ion transport
A0008076cellular_componentvoltage-gated potassium channel complex
A0016020cellular_componentmembrane
A0051260biological_processprotein homooligomerization
A0055085biological_processtransmembrane transport
B0005216molecular_functionmonoatomic ion channel activity
B0005249molecular_functionvoltage-gated potassium channel activity
B0006811biological_processmonoatomic ion transport
B0006813biological_processpotassium ion transport
B0008076cellular_componentvoltage-gated potassium channel complex
B0016020cellular_componentmembrane
B0051260biological_processprotein homooligomerization
B0055085biological_processtransmembrane transport
C0005216molecular_functionmonoatomic ion channel activity
C0005249molecular_functionvoltage-gated potassium channel activity
C0006811biological_processmonoatomic ion transport
C0006813biological_processpotassium ion transport
C0008076cellular_componentvoltage-gated potassium channel complex
C0016020cellular_componentmembrane
C0051260biological_processprotein homooligomerization
C0055085biological_processtransmembrane transport
D0005216molecular_functionmonoatomic ion channel activity
D0005249molecular_functionvoltage-gated potassium channel activity
D0006811biological_processmonoatomic ion transport
D0006813biological_processpotassium ion transport
D0008076cellular_componentvoltage-gated potassium channel complex
D0016020cellular_componentmembrane
D0051260biological_processprotein homooligomerization
D0055085biological_processtransmembrane transport
I0001508biological_processaction potential
I0005250molecular_functionA-type (transient outward) potassium channel activity
I0005267molecular_functionpotassium channel activity
I0005509molecular_functioncalcium ion binding
I0005513biological_processdetection of calcium ion
I0005515molecular_functionprotein binding
I0005737cellular_componentcytoplasm
I0005886cellular_componentplasma membrane
I0006813biological_processpotassium ion transport
I0006936biological_processmuscle contraction
I0007165biological_processsignal transduction
I0007268biological_processchemical synaptic transmission
I0008016biological_processregulation of heart contraction
I0008076cellular_componentvoltage-gated potassium channel complex
I0015459molecular_functionpotassium channel regulator activity
I0030425cellular_componentdendrite
I0034702cellular_componentmonoatomic ion channel complex
I0034705cellular_componentpotassium channel complex
I0044325molecular_functiontransmembrane transporter binding
I0044877molecular_functionprotein-containing complex binding
I0045163biological_processclustering of voltage-gated potassium channels
I0045202cellular_componentsynapse
I0046872molecular_functionmetal ion binding
I0046923molecular_functionER retention sequence binding
I0071193cellular_componentKv4.2-KChIP2 channel complex
I0071805biological_processpotassium ion transmembrane transport
I0086008molecular_functionvoltage-gated potassium channel activity involved in cardiac muscle cell action potential repolarization
I0086009biological_processmembrane repolarization
I0086013biological_processmembrane repolarization during cardiac muscle cell action potential
I0097623biological_processpotassium ion export across plasma membrane
I1901379biological_processregulation of potassium ion transmembrane transport
I1903766biological_processpositive regulation of potassium ion export across plasma membrane
I1903818biological_processpositive regulation of voltage-gated potassium channel activity
J0001508biological_processaction potential
J0005250molecular_functionA-type (transient outward) potassium channel activity
J0005267molecular_functionpotassium channel activity
J0005509molecular_functioncalcium ion binding
J0005513biological_processdetection of calcium ion
J0005515molecular_functionprotein binding
J0005737cellular_componentcytoplasm
J0005886cellular_componentplasma membrane
J0006813biological_processpotassium ion transport
J0006936biological_processmuscle contraction
J0007165biological_processsignal transduction
J0007268biological_processchemical synaptic transmission
J0008016biological_processregulation of heart contraction
J0008076cellular_componentvoltage-gated potassium channel complex
J0015459molecular_functionpotassium channel regulator activity
J0030425cellular_componentdendrite
J0034702cellular_componentmonoatomic ion channel complex
J0034705cellular_componentpotassium channel complex
J0044325molecular_functiontransmembrane transporter binding
J0044877molecular_functionprotein-containing complex binding
J0045163biological_processclustering of voltage-gated potassium channels
J0045202cellular_componentsynapse
J0046872molecular_functionmetal ion binding
J0046923molecular_functionER retention sequence binding
J0071193cellular_componentKv4.2-KChIP2 channel complex
J0071805biological_processpotassium ion transmembrane transport
J0086008molecular_functionvoltage-gated potassium channel activity involved in cardiac muscle cell action potential repolarization
J0086009biological_processmembrane repolarization
J0086013biological_processmembrane repolarization during cardiac muscle cell action potential
J0097623biological_processpotassium ion export across plasma membrane
J1901379biological_processregulation of potassium ion transmembrane transport
J1903766biological_processpositive regulation of potassium ion export across plasma membrane
J1903818biological_processpositive regulation of voltage-gated potassium channel activity
K0001508biological_processaction potential
K0005250molecular_functionA-type (transient outward) potassium channel activity
K0005267molecular_functionpotassium channel activity
K0005509molecular_functioncalcium ion binding
K0005513biological_processdetection of calcium ion
K0005515molecular_functionprotein binding
K0005737cellular_componentcytoplasm
K0005886cellular_componentplasma membrane
K0006813biological_processpotassium ion transport
K0006936biological_processmuscle contraction
K0007165biological_processsignal transduction
K0007268biological_processchemical synaptic transmission
K0008016biological_processregulation of heart contraction
K0008076cellular_componentvoltage-gated potassium channel complex
K0015459molecular_functionpotassium channel regulator activity
K0030425cellular_componentdendrite
K0034702cellular_componentmonoatomic ion channel complex
K0034705cellular_componentpotassium channel complex
K0044325molecular_functiontransmembrane transporter binding
K0044877molecular_functionprotein-containing complex binding
K0045163biological_processclustering of voltage-gated potassium channels
K0045202cellular_componentsynapse
K0046872molecular_functionmetal ion binding
K0046923molecular_functionER retention sequence binding
K0071193cellular_componentKv4.2-KChIP2 channel complex
K0071805biological_processpotassium ion transmembrane transport
K0086008molecular_functionvoltage-gated potassium channel activity involved in cardiac muscle cell action potential repolarization
K0086009biological_processmembrane repolarization
K0086013biological_processmembrane repolarization during cardiac muscle cell action potential
K0097623biological_processpotassium ion export across plasma membrane
K1901379biological_processregulation of potassium ion transmembrane transport
K1903766biological_processpositive regulation of potassium ion export across plasma membrane
K1903818biological_processpositive regulation of voltage-gated potassium channel activity
L0001508biological_processaction potential
L0005250molecular_functionA-type (transient outward) potassium channel activity
L0005267molecular_functionpotassium channel activity
L0005509molecular_functioncalcium ion binding
L0005513biological_processdetection of calcium ion
L0005515molecular_functionprotein binding
L0005737cellular_componentcytoplasm
L0005886cellular_componentplasma membrane
L0006813biological_processpotassium ion transport
L0006936biological_processmuscle contraction
L0007165biological_processsignal transduction
L0007268biological_processchemical synaptic transmission
L0008016biological_processregulation of heart contraction
L0008076cellular_componentvoltage-gated potassium channel complex
L0015459molecular_functionpotassium channel regulator activity
L0030425cellular_componentdendrite
L0034702cellular_componentmonoatomic ion channel complex
L0034705cellular_componentpotassium channel complex
L0044325molecular_functiontransmembrane transporter binding
L0044877molecular_functionprotein-containing complex binding
L0045163biological_processclustering of voltage-gated potassium channels
L0045202cellular_componentsynapse
L0046872molecular_functionmetal ion binding
L0046923molecular_functionER retention sequence binding
L0071193cellular_componentKv4.2-KChIP2 channel complex
L0071805biological_processpotassium ion transmembrane transport
L0086008molecular_functionvoltage-gated potassium channel activity involved in cardiac muscle cell action potential repolarization
L0086009biological_processmembrane repolarization
L0086013biological_processmembrane repolarization during cardiac muscle cell action potential
L0097623biological_processpotassium ion export across plasma membrane
L1901379biological_processregulation of potassium ion transmembrane transport
L1903766biological_processpositive regulation of potassium ion export across plasma membrane
L1903818biological_processpositive regulation of voltage-gated potassium channel activity
Functional Information from PROSITE/UniProt
site_idPS00018
Number of Residues13
DetailsEF_HAND_1 EF-hand calcium-binding domain. DTNHDGSVSfeDF
ChainResidueDetails
IASP135-PHE147
IASP171-MET183
IASP219-PHE231

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues56
DetailsBINDING: BINDING => ECO:0000255|PROSITE-ProRule:PRU00448
ChainResidueDetails
IVAL153
IPRO200
ILYS237
IGLU239
IILE241
IPHE248
JVAL153
JLEU155
JGLY157
JVAL159
JASN164
ILEU155
JSER189
JTYR191
JMET193
JGLY195
JPRO200
JLYS237
JGLU239
JILE241
JPHE248
KVAL153
IGLY157
KLEU155
KGLY157
KVAL159
KASN164
KSER189
KTYR191
KMET193
KGLY195
KPRO200
KLYS237
IVAL159
KGLU239
KILE241
KPHE248
LVAL153
LLEU155
LGLY157
LVAL159
LASN164
LSER189
LTYR191
IASN164
LMET193
LGLY195
LPRO200
LLYS237
LGLU239
LILE241
LPHE248
ISER189
ITYR191
IMET193
IGLY195

site_idSWS_FT_FI2
Number of Residues4
DetailsMOD_RES: Phosphoserine => ECO:0000250|UniProtKB:Q9JM59
ChainResidueDetails
ISER9
JSER9
KSER9
LSER9

site_idSWS_FT_FI3
Number of Residues8
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250|UniProtKB:Q9JM59
ChainResidueDetails
ICYS45
CTHR280-SER286
CTYR344-ILE357
CPRO378-LYS384
DGLU205-ALA228
DTHR280-SER286
DTYR344-ILE357
DPRO378-LYS384
ICYS46
JCYS45
JCYS46
KCYS45
KCYS46
LCYS45
LCYS46
CGLU205-ALA228

site_idSWS_FT_FI4
Number of Residues84
DetailsTRANSMEM: Helical; Name=Segment S2 => ECO:0000250|UniProtKB:P63142
ChainResidueDetails
APHE229-ALA250
BPHE229-ALA250
CPHE229-ALA250
DPHE229-ALA250

site_idSWS_FT_FI5
Number of Residues68
DetailsTRANSMEM: Helical; Name=Segment S3 => ECO:0000250|UniProtKB:P63142
ChainResidueDetails
AMET262-MET279
BMET262-MET279
CMET262-MET279
DMET262-MET279

site_idSWS_FT_FI6
Number of Residues76
DetailsTRANSMEM: Helical; Voltage-sensor; Name=Segment S4 => ECO:0000250|UniProtKB:P63142
ChainResidueDetails
AGLY287-HIS306
BGLY287-HIS306
CGLY287-HIS306
DGLY287-HIS306

site_idSWS_FT_FI7
Number of Residues84
DetailsTRANSMEM: Helical; Name=Segment S5 => ECO:0000250|UniProtKB:P63142
ChainResidueDetails
ASER322-PHE343
BSER322-PHE343
CSER322-PHE343
DSER322-PHE343

site_idSWS_FT_FI8
Number of Residues44
DetailsINTRAMEM: Helical; Name=Pore helix => ECO:0000250|UniProtKB:P63142
ChainResidueDetails
APRO358-THR369
BPRO358-THR369
CPRO358-THR369
DPRO358-THR369

site_idSWS_FT_FI9
Number of Residues28
DetailsINTRAMEM: INTRAMEM => ECO:0000250|UniProtKB:P63142
ChainResidueDetails
ATHR370-VAL377
BTHR370-VAL377
CTHR370-VAL377
DTHR370-VAL377

site_idSWS_FT_FI10
Number of Residues112
DetailsTRANSMEM: Helical; Name=Segment S6 => ECO:0000250|UniProtKB:P63142
ChainResidueDetails
AILE385-TYR413
BILE385-TYR413
CILE385-TYR413
DILE385-TYR413

site_idSWS_FT_FI11
Number of Residues12
DetailsBINDING: BINDING => ECO:0000250|UniProtKB:Q63881
ChainResidueDetails
AHIS105
DHIS105
DCYS132
DCYS133
ACYS132
ACYS133
BHIS105
BCYS132
BCYS133
CHIS105
CCYS132
CCYS133

site_idSWS_FT_FI12
Number of Residues4
DetailsMOD_RES: Phosphothreonine => ECO:0000250|UniProtKB:Q63881
ChainResidueDetails
ATHR38
BTHR38
CTHR38
DTHR38

site_idSWS_FT_FI13
Number of Residues4
DetailsMOD_RES: Phosphoserine => ECO:0000250|UniProtKB:Q63881
ChainResidueDetails
ASER438
BSER438
CSER438
DSER438

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PDB entries from 2024-07-10

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