7UBO
Crystal Structure of the first bromodomain of human BRDT in complex with the inhibitor CCD-956
Functional Information from PROSITE/UniProt
site_id | PS00633 |
Number of Residues | 60 |
Details | BROMODOMAIN_1 Bromodomain signature. SwpFqrpvDavklqlpDYYtiIknpMdlntIkkrlenky..Yakaseciedfnt.MfsNCylY |
Chain | Residue | Details |
A | SER49-TYR108 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 4 |
Details | BINDING: BINDING => ECO:0000269|PubMed:22901802, ECO:0007744|PDB:4FLP |
Chain | Residue | Details |
A | ASN109 | |
B | ASN109 | |
C | ASN109 | |
D | ASN109 |
site_id | SWS_FT_FI2 |
Number of Residues | 8 |
Details | SITE: Histone H4K5ac binding => ECO:0000250|UniProtKB:Q91Y44 |
Chain | Residue | Details |
A | ASN109 | |
A | ASP114 | |
B | ASN109 | |
B | ASP114 | |
C | ASN109 | |
C | ASP114 | |
D | ASN109 | |
D | ASP114 |