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7UBO

Crystal Structure of the first bromodomain of human BRDT in complex with the inhibitor CCD-956

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SwpFqrpvDavklqlpDYYtiIknpMdlntIkkrlenky..Yakaseciedfnt.MfsNCylY
ChainResidueDetails
ASER49-TYR108

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues4
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"22901802","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"4FLP","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsSite: {"description":"Histone H4K5ac binding","evidences":[{"source":"UniProtKB","id":"Q91Y44","evidenceCode":"ECO:0000250"}]}
ChainResidueDetails

247947

PDB entries from 2026-01-21

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