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7QVM

Human Oxytocin receptor (OTR) oxytocin Gq chimera (mGoqi) complex

Functional Information from GO Data
ChainGOidnamespacecontents
A0003924molecular_functionGTPase activity
A0005525molecular_functionGTP binding
A0007186biological_processG protein-coupled receptor signaling pathway
A0007188biological_processadenylate cyclase-modulating G protein-coupled receptor signaling pathway
A0019001molecular_functionguanyl nucleotide binding
A0031683molecular_functionG-protein beta/gamma-subunit complex binding
B0001750cellular_componentphotoreceptor outer segment
B0003924molecular_functionGTPase activity
B0005515molecular_functionprotein binding
B0005737cellular_componentcytoplasm
B0005765cellular_componentlysosomal membrane
B0005829cellular_componentcytosol
B0005834cellular_componentheterotrimeric G-protein complex
B0005886cellular_componentplasma membrane
B0007165biological_processsignal transduction
B0007186biological_processG protein-coupled receptor signaling pathway
B0007191biological_processadenylate cyclase-activating dopamine receptor signaling pathway
B0007200biological_processphospholipase C-activating G protein-coupled receptor signaling pathway
B0007213biological_processG protein-coupled acetylcholine receptor signaling pathway
B0007265biological_processRas protein signal transduction
B0008283biological_processcell population proliferation
B0016020cellular_componentmembrane
B0030159molecular_functionsignaling receptor complex adaptor activity
B0044877molecular_functionprotein-containing complex binding
B0045202cellular_componentsynapse
B0050909biological_processsensory perception of taste
B0051020molecular_functionGTPase binding
B0060041biological_processretina development in camera-type eye
B0070062cellular_componentextracellular exosome
B0071380biological_processcellular response to prostaglandin E stimulus
B0071870biological_processcellular response to catecholamine stimulus
B0097381cellular_componentphotoreceptor disc membrane
B1903561cellular_componentextracellular vesicle
G0005515molecular_functionprotein binding
G0005834cellular_componentheterotrimeric G-protein complex
G0005886cellular_componentplasma membrane
G0007165biological_processsignal transduction
G0007186biological_processG protein-coupled receptor signaling pathway
G0007191biological_processadenylate cyclase-activating dopamine receptor signaling pathway
G0016020cellular_componentmembrane
G0031681molecular_functionG-protein beta-subunit binding
G0048144biological_processfibroblast proliferation
G0070062cellular_componentextracellular exosome
G0071380biological_processcellular response to prostaglandin E stimulus
G0071870biological_processcellular response to catecholamine stimulus
L0005185molecular_functionneurohypophyseal hormone activity
L0005576cellular_componentextracellular region
R0001967biological_processsuckling behavior
R0001975biological_processresponse to amphetamine
R0001992biological_processregulation of systemic arterial blood pressure by vasopressin
R0004930molecular_functionG protein-coupled receptor activity
R0004990molecular_functionoxytocin receptor activity
R0005000molecular_functionvasopressin receptor activity
R0005886cellular_componentplasma membrane
R0005902cellular_componentmicrovillus
R0005912cellular_componentadherens junction
R0006936biological_processmuscle contraction
R0007166biological_processcell surface receptor signaling pathway
R0007186biological_processG protein-coupled receptor signaling pathway
R0007204biological_processpositive regulation of cytosolic calcium ion concentration
R0007507biological_processheart development
R0007565biological_processfemale pregnancy
R0007595biological_processlactation
R0007613biological_processmemory
R0009410biological_processresponse to xenobiotic stimulus
R0010701biological_processpositive regulation of norepinephrine secretion
R0014070biological_processresponse to organic cyclic compound
R0016020cellular_componentmembrane
R0016324cellular_componentapical plasma membrane
R0017046molecular_functionpeptide hormone binding
R0021537biological_processtelencephalon development
R0032230biological_processpositive regulation of synaptic transmission, GABAergic
R0032355biological_processresponse to estradiol
R0032570biological_processresponse to progesterone
R0032870biological_processcellular response to hormone stimulus
R0034059biological_processresponse to anoxia
R0034097biological_processresponse to cytokine
R0035176biological_processsocial behavior
R0042220biological_processresponse to cocaine
R0042277molecular_functionpeptide binding
R0042711biological_processmaternal behavior
R0042713biological_processsperm ejaculation
R0042755biological_processeating behavior
R0043434biological_processresponse to peptide hormone
R0044849biological_processestrous cycle
R0045777biological_processpositive regulation of blood pressure
R0045907biological_processpositive regulation of vasoconstriction
R0048545biological_processresponse to steroid hormone
R0048565biological_processdigestive tract development
R0051965biological_processpositive regulation of synapse assembly
R0051968biological_processpositive regulation of synaptic transmission, glutamatergic
R0060137biological_processmaternal process involved in parturition
R0060406biological_processpositive regulation of penile erection
R0070371biological_processERK1 and ERK2 cascade
R0070474biological_processpositive regulation of uterine smooth muscle contraction
R0120162biological_processpositive regulation of cold-induced thermogenesis
Functional Information from PROSITE/UniProt
site_idPS00237
Number of Residues17
DetailsG_PROTEIN_RECEP_F1_1 G-protein coupled receptors family 1 signature. ASTyLLLLMSLDRCLaI
ChainResidueDetails
RALA125-ILE141

site_idPS00264
Number of Residues9
DetailsNEUROHYPOPHYS_HORM Neurohypophysial hormones signature. CYIqNCPlG
ChainResidueDetails
LCYS1-GLY9

site_idPS00678
Number of Residues15
DetailsWD_REPEATS_1 Trp-Asp (WD) repeats signature. LVSAsqDgKLIIWDS
ChainResidueDetails
BLEU70-SER84
BILE157-ILE171
BLEU285-ALA299

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues92
DetailsTOPO_DOM: Extracellular => ECO:0000255
ChainResidueDetails
RMET1-LEU38
RLEU98-ARG113
RSER176-THR202
RGLN295-SER309
AASN270
AALA326

site_idSWS_FT_FI2
Number of Residues24
DetailsTRANSMEM: Helical; Name=1 => ECO:0000255
ChainResidueDetails
RALA39-ALA63

site_idSWS_FT_FI3
Number of Residues77
DetailsTOPO_DOM: Cytoplasmic => ECO:0000255
ChainResidueDetails
RLEU64-LEU74
RASP136-ARG154
RLYS226-LYS275

site_idSWS_FT_FI4
Number of Residues22
DetailsTRANSMEM: Helical; Name=2 => ECO:0000255
ChainResidueDetails
RPHE75-LEU97

site_idSWS_FT_FI5
Number of Residues21
DetailsTRANSMEM: Helical; Name=3 => ECO:0000255
ChainResidueDetails
RLEU114-LEU135

site_idSWS_FT_FI6
Number of Residues20
DetailsTRANSMEM: Helical; Name=4 => ECO:0000255
ChainResidueDetails
RLEU155-PHE175

site_idSWS_FT_FI7
Number of Residues22
DetailsTRANSMEM: Helical; Name=5 => ECO:0000255
ChainResidueDetails
RTRP203-PHE225

site_idSWS_FT_FI8
Number of Residues18
DetailsTRANSMEM: Helical; Name=6 => ECO:0000255
ChainResidueDetails
RMET276-VAL294

site_idSWS_FT_FI9
Number of Residues22
DetailsTRANSMEM: Helical; Name=7 => ECO:0000255
ChainResidueDetails
RALA310-PHE332

site_idSWS_FT_FI10
Number of Residues3
DetailsCARBOHYD: N-linked (GlcNAc...) asparagine => ECO:0000255
ChainResidueDetails
RASN8
RASN15
RASN26

222926

PDB entries from 2024-07-24

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