Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

7OFE

Keap1 kelch domain bound to a small molecule inhibitor of the Keap1-Nrf2 protein-protein interaction

Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue SO4 A 701
ChainResidue
AILE435
AHIS437
ASER438
ASER439
AARG494
AHOH814
AHOH871
AHOH901
AHOH987

site_idAC2
Number of Residues6
Detailsbinding site for residue SO4 A 702
ChainResidue
ACYS434
AHIS436
AARG459
AARG494
AARG498
AHOH830

site_idAC3
Number of Residues5
Detailsbinding site for residue DMS A 703
ChainResidue
AARG380
AASN382
AASN414
ADMS705
AHOH801

site_idAC4
Number of Residues3
Detailsbinding site for residue DMS A 704
ChainResidue
AHIS451
ALEU452
AHOH803

site_idAC5
Number of Residues5
Detailsbinding site for residue DMS A 705
ChainResidue
ATYR334
AARG415
ASER602
AGLY603
ADMS703

site_idAC6
Number of Residues2
Detailsbinding site for residue DMS A 706
ChainResidue
AARG494
AASN495

site_idAC7
Number of Residues3
Detailsbinding site for residue DMS A 707
ChainResidue
ALEU457
AARG459
AHOH888

site_idAC8
Number of Residues7
Detailsbinding site for residue DMS A 708
ChainResidue
ATHR388
AASP389
ASER390
ASER391
AARG470
AHOH820
AHOH855

site_idAC9
Number of Residues1
Detailsbinding site for residue DMS A 709
ChainResidue
AARG442

site_idAD1
Number of Residues10
Detailsbinding site for residue VBQ A 710
ChainResidue
AARG415
AARG483
ASER508
AGLY509
ATYR525
AGLN530
ASER555
ATYR572
APHE577
ASER602

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Sensor for electrophilic agents => ECO:0000269|PubMed:20498371
ChainResidueDetails
ACYS434

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: S-cGMP-cysteine => ECO:0000269|PubMed:20498371
ChainResidueDetails
ACYS434

site_idSWS_FT_FI3
Number of Residues1
DetailsMOD_RES: S-(2-succinyl)cysteine => ECO:0000269|PubMed:22014577
ChainResidueDetails
ACYS613

222415

PDB entries from 2024-07-10

PDB statisticsPDBj update infoContact PDBjnumon