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7OFD

Keap1 kelch domain bound to a small molecule fragment

Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue SO4 A 701
ChainResidue
AILE435
AHIS437
ASER438
ASER439
AARG494
AHOH815
AHOH826
AHOH878
AHOH948

site_idAC2
Number of Residues6
Detailsbinding site for residue SO4 A 702
ChainResidue
ACYS434
AHIS436
AARG459
AARG494
AARG498
AHOH854

site_idAC3
Number of Residues5
Detailsbinding site for residue DMS A 703
ChainResidue
AARG380
AASN382
AASN414
AVBW714
AHOH801

site_idAC4
Number of Residues2
Detailsbinding site for residue DMS A 704
ChainResidue
AHIS451
ALEU452

site_idAC5
Number of Residues3
Detailsbinding site for residue DMS A 705
ChainResidue
AARG494
AASN495
ADMS712

site_idAC6
Number of Residues3
Detailsbinding site for residue DMS A 706
ChainResidue
AMET456
ALEU457
AARG459

site_idAC7
Number of Residues7
Detailsbinding site for residue DMS A 707
ChainResidue
ATHR388
AASP389
ASER390
ASER391
AARG470
AHOH827
AHOH862

site_idAC8
Number of Residues2
Detailsbinding site for residue DMS A 708
ChainResidue
AHIS424
AARG442

site_idAC9
Number of Residues3
Detailsbinding site for residue DMS A 709
ChainResidue
APRO361
AHIS553
AHOH946

site_idAD1
Number of Residues4
Detailsbinding site for residue DMS A 710
ChainResidue
AARG354
ALEU355
AASP357
AHIS552

site_idAD2
Number of Residues5
Detailsbinding site for residue DMS A 711
ChainResidue
ATYR525
AGLN530
ASER555
ATYR572
AVBW714

site_idAD3
Number of Residues5
Detailsbinding site for residue DMS A 712
ChainResidue
ALEU452
AVAL453
AALA454
AASN495
ADMS705

site_idAD4
Number of Residues6
Detailsbinding site for residue DMS A 713
ChainResidue
AARG380
AGLY433
AVAL539
AGLU540
AHOH879
AHOH956

site_idAD5
Number of Residues6
Detailsbinding site for residue VBW A 714
ChainResidue
ATYR334
ASER363
AALA556
ASER602
ADMS703
ADMS711

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues45
DetailsRepeat: {"description":"Kelch 1"}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues50
DetailsRepeat: {"description":"Kelch 2"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues46
DetailsRepeat: {"description":"Kelch 3"}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues46
DetailsRepeat: {"description":"Kelch 4"}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues45
DetailsRepeat: {"description":"Kelch 5"}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues46
DetailsRepeat: {"description":"Kelch 6"}
ChainResidueDetails

site_idSWS_FT_FI7
Number of Residues1
DetailsSite: {"description":"Sensor for electrophilic agents","evidences":[{"source":"PubMed","id":"20498371","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI8
Number of Residues1
DetailsModified residue: {"description":"S-cGMP-cysteine","evidences":[{"source":"PubMed","id":"20498371","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI9
Number of Residues1
DetailsModified residue: {"description":"S-(2-succinyl)cysteine","evidences":[{"source":"PubMed","id":"22014577","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

246031

PDB entries from 2025-12-10

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