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7NDO

ER-PRS*(-) (L536S, L372R) in complex with raloxifene

Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue RAL A 601
ChainResidue
ALEU346
AASN532
APRO535
AHOH761
AALA350
AASP351
AGLU353
ALEU354
ALEU387
AARG394
AILE424
AHIS524

site_idAC2
Number of Residues4
Detailsbinding site for residue EDO A 602
ChainResidue
AASP407
ALEU409
AGLN414
AHOH714

site_idAC3
Number of Residues4
Detailsbinding site for residue EDO A 603
ChainResidue
AARG372
AEDO604
AHOH750
AHOH770

site_idAC4
Number of Residues7
Detailsbinding site for residue EDO A 604
ChainResidue
ALYS362
AARG372
ALEU544
AEDO603
AHOH725
BVAL368
BASP369

site_idAC5
Number of Residues5
Detailsbinding site for residue CL A 605
ChainResidue
ATYR328
AARG352
AHOH789
BHIS356
BHOH778

site_idAC6
Number of Residues4
Detailsbinding site for residue CL A 606
ChainResidue
AHIS356
AHOH755
AHOH789
BTYR328

site_idAC7
Number of Residues1
Detailsbinding site for residue CL A 607
ChainResidue
AGLU444

site_idAC8
Number of Residues12
Detailsbinding site for residue RAL B 601
ChainResidue
BLEU346
BTHR347
BASP351
BGLU353
BLEU387
BARG394
BILE424
BHIS524
BVAL533
BPRO535
BHOH704
BHOH748

site_idAC9
Number of Residues11
Detailsbinding site for residue EDO B 602
ChainResidue
BASP313
BILE316
BSER317
BLEU320
BGLU339
BTRP488
BLYS492
BEDO604
BHOH702
BHOH705
BHOH735

site_idAD1
Number of Residues6
Detailsbinding site for residue EDO B 603
ChainResidue
BGLU323
BARG394
BPHE445
BLYS449
BHOH718
BHOH743

site_idAD2
Number of Residues7
Detailsbinding site for residue EDO B 604
ChainResidue
BSER317
BLEU320
BGLU321
BEDO602
BHOH705
BHOH706
BHOH715

site_idAD3
Number of Residues5
Detailsbinding site for residue EDO B 605
ChainResidue
BASP407
BLEU408
BLEU409
BGLN414
BTHR465

site_idAD4
Number of Residues6
Detailsbinding site for residue EDO B 606
ChainResidue
BGLN441
BGLU444
BTYR489
BSER493
BLEU495
BARG503

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:9338790, ECO:0000269|PubMed:9600906, ECO:0007744|PDB:1A52, ECO:0007744|PDB:1ERE
ChainResidueDetails
AGLU353
AARG394
AHIS524
BGLU353
BARG394
BHIS524

site_idSWS_FT_FI2
Number of Residues2
DetailsMOD_RES: Phosphotyrosine; by Tyr-kinases => ECO:0000269|PubMed:7539106
ChainResidueDetails
ATYR537
BTYR537

site_idSWS_FT_FI3
Number of Residues2
DetailsLIPID: S-palmitoyl cysteine => ECO:0000250
ChainResidueDetails
ACYS447
BCYS447

224201

PDB entries from 2024-08-28

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