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7LZR

Crystal structure of the BCL6 BTB domain in complex with OICR-10256

Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue SO4 A 201
ChainResidue
AARG26
ASER27
AASP29
AARG44
DASP29
DARG44

site_idAC2
Number of Residues7
Detailsbinding site for residue GOL A 202
ChainResidue
ATHR92
AHOH301
DSER27
DARG28
AASN23
AARG26
AASP88

site_idAC3
Number of Residues1
Detailsbinding site for residue CL A 203
ChainResidue
AASN73

site_idAC4
Number of Residues24
Detailsbinding site for residue YJJ A 204
ChainResidue
AMET51
AALA52
ACYS53
ASER54
AGLY55
ATYR58
APHE89
AGLN113
AMET114
AGLU115
AHIS116
AVAL117
AHOH315
AHOH324
BHIS14
BASP17
BASN21
BARG24
BLEU25
BARG28
CGLU81
CILE85
CASN96
CARG98

site_idAC5
Number of Residues7
Detailsbinding site for residue GOL A 205
ChainResidue
ALEU31
AASP33
ALYS47
ATHR48
BASP33
BLYS47
BTHR48

site_idAC6
Number of Residues21
Detailsbinding site for residue YJJ B 201
ChainResidue
AHIS14
AASP17
AARG24
ALEU25
AARG28
BMET51
BALA52
BCYS53
BSER54
BGLY55
BTYR58
BPHE89
BGLN113
BMET114
BGLU115
BHIS116
BVAL117
BHOH319
BHOH329
BHOH337
DHOH372

site_idAC7
Number of Residues7
Detailsbinding site for residue SO4 B 202
ChainResidue
AASP75
AILE78
AHOH344
BASP75
BGLU77
BILE78
BHOH322

site_idAC8
Number of Residues3
Detailsbinding site for residue CL B 203
ChainResidue
BARG98
BGLU99
BGLY100

site_idAC9
Number of Residues1
Detailsbinding site for residue CL B 204
ChainResidue
BTHR12

site_idAD1
Number of Residues4
Detailsbinding site for residue SO4 C 201
ChainResidue
CPHE11
CTHR12
CARG13
DHIS116

site_idAD2
Number of Residues6
Detailsbinding site for residue GOL C 202
ChainResidue
CASP33
CLYS47
CTHR48
DASP33
DLYS47
DTHR48

site_idAD3
Number of Residues20
Detailsbinding site for residue YJJ C 203
ChainResidue
CVAL117
CHOH323
CHOH331
CHOH340
DHIS14
DASP17
DARG24
DLEU25
AASN96
CMET51
CALA52
CCYS53
CSER54
CGLY55
CTYR58
CPHE89
CGLN113
CMET114
CGLU115
CHIS116

site_idAD4
Number of Residues2
Detailsbinding site for residue CL C 204
ChainResidue
CARG67
DLEU31

site_idAD5
Number of Residues26
Detailsbinding site for residue YJJ D 201
ChainResidue
BGLU41
BPHE43
BGLU81
BHOH303
CHIS14
CASP17
CASN21
CARG24
CLEU25
CARG28
DMET51
DALA52
DCYS53
DSER54
DGLY55
DTYR58
DPHE89
DGLN113
DMET114
DGLU115
DHIS116
DVAL117
DHOH314
DHOH328
DHOH337
DHOH345

site_idAD6
Number of Residues7
Detailsbinding site for residue SO4 D 202
ChainResidue
CHIS116
CHOH319
DGLN10
DPHE11
DTHR12
DARG13
DHOH316

site_idAD7
Number of Residues6
Detailsbinding site for residue SO4 D 203
ChainResidue
DTHR32
DASP33
DVAL34
DVAL35
DARG44
DSER70

site_idAD8
Number of Residues1
Detailsbinding site for residue CL D 204
ChainResidue
DLYS66

220472

PDB entries from 2024-05-29

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