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7LGK

Crystal structure of soluble guanylate cyclase activator runcaciguat (BAY 1101042) bound to nostoc H-NOX domain

Functional Information from GO Data
ChainGOidnamespacecontents
A0020037molecular_functionheme binding
A0046872molecular_functionmetal ion binding
B0020037molecular_functionheme binding
B0046872molecular_functionmetal ion binding
Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue XZ7 A 1001
ChainResidue
AMET1
ATYR134
ASER136
AARG138
ALEU141
AMET144
ALEU148
AGOL1003
ATRP74
ATHR78
ATYR83
ALEU101
AHIS105
ALEU115
APRO118
APHE120

site_idAC2
Number of Residues3
Detailsbinding site for residue CL A 1002
ChainResidue
AARG116
AARG138
AGOL1004

site_idAC3
Number of Residues2
Detailsbinding site for residue GOL A 1003
ChainResidue
AXZ71001
AHOH1130

site_idAC4
Number of Residues7
Detailsbinding site for residue GOL A 1004
ChainResidue
AMET1
ATYR43
AASP45
AGLN114
AARG116
AARG138
ACL1002

site_idAC5
Number of Residues4
Detailsbinding site for residue GOL A 1005
ChainResidue
AHIS16
AHIS17
ALYS61
BLYS128

site_idAC6
Number of Residues16
Detailsbinding site for residue XZ7 B 1001
ChainResidue
BTRP74
BTHR78
BTYR83
BLEU101
BHIS105
BLEU115
BPRO118
BPHE120
BTYR134
BSER136
BARG138
BLEU141
BMET144
BLEU148
BGOL1004
BHOH1121

site_idAC7
Number of Residues4
Detailsbinding site for residue CL B 1002
ChainResidue
BARG116
BARG138
BGOL1003
BHOH1102

site_idAC8
Number of Residues7
Detailsbinding site for residue GOL B 1003
ChainResidue
BMET1
BALA42
BTYR43
BGLN114
BARG116
BARG138
BCL1002

site_idAC9
Number of Residues3
Detailsbinding site for residue GOL B 1004
ChainResidue
BVAL108
BXZ71001
BHOH1102

site_idAD1
Number of Residues5
Detailsbinding site for residue GOL B 1005
ChainResidue
BGLY82
BSER89
BHOH1106
BHOH1118
BHOH1119

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PDB entries from 2024-07-10

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