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7LEJ

Crystal structure of the second bromodomain (BD2) of human BRDT bound to Volasertib

Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue IBI A 401
ChainResidue
ATYR259
AHIS356
AHOH508
AHOH530
AALA263
APRO294
AVAL299
AALA303
ALEU304
ALEU306
ATYR309
AASN352

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFynpvDvnalglhNYYdvVknpMdlgtIkekmdnqe..Ykdaykfaadvrl.MfmNCykY
ChainResidueDetails
AALA292-TYR351

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues109
DetailsDomain: {"description":"Bromo 2","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

249697

PDB entries from 2026-02-25

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