7LEJ
Crystal structure of the second bromodomain (BD2) of human BRDT bound to Volasertib
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 12 |
Details | binding site for residue IBI A 401 |
Chain | Residue |
A | TYR259 |
A | HIS356 |
A | HOH508 |
A | HOH530 |
A | ALA263 |
A | PRO294 |
A | VAL299 |
A | ALA303 |
A | LEU304 |
A | LEU306 |
A | TYR309 |
A | ASN352 |
Functional Information from PROSITE/UniProt
site_id | PS00633 |
Number of Residues | 60 |
Details | BROMODOMAIN_1 Bromodomain signature. AwpFynpvDvnalglhNYYdvVknpMdlgtIkekmdnqe..Ykdaykfaadvrl.MfmNCykY |
Chain | Residue | Details |
A | ALA292-TYR351 |