7LAJ
Crystal structure of the first bromodomain (BD1) of human BRD2 bound to Ro3280
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 15 |
Details | binding site for residue 79C A 201 |
Chain | Residue |
A | PRO98 |
A | LEU187 |
A | THR190 |
A | HOH308 |
A | HOH321 |
A | HOH327 |
A | HOH348 |
A | PHE99 |
A | VAL103 |
A | LEU110 |
A | TYR113 |
A | TYR155 |
A | ASN156 |
A | GLN185 |
A | GLU186 |
Functional Information from PROSITE/UniProt
site_id | PS00633 |
Number of Residues | 60 |
Details | BROMODOMAIN_1 Bromodomain signature. AwpFrqpvDavklglpDYHkiIkqpMdmgtIkrrlenny..Ywaasecmqdfnt.MftNCyiY |
Chain | Residue | Details |
A | ALA96-TYR155 |