7LAJ
Crystal structure of the first bromodomain (BD1) of human BRD2 bound to Ro3280
Functional Information from PDB Data
| site_id | AC1 |
| Number of Residues | 15 |
| Details | binding site for residue 79C A 201 |
| Chain | Residue |
| A | PRO98 |
| A | LEU187 |
| A | THR190 |
| A | HOH308 |
| A | HOH321 |
| A | HOH327 |
| A | HOH348 |
| A | PHE99 |
| A | VAL103 |
| A | LEU110 |
| A | TYR113 |
| A | TYR155 |
| A | ASN156 |
| A | GLN185 |
| A | GLU186 |
Functional Information from PROSITE/UniProt
| site_id | PS00633 |
| Number of Residues | 60 |
| Details | BROMODOMAIN_1 Bromodomain signature. AwpFrqpvDavklglpDYHkiIkqpMdmgtIkrrlenny..Ywaasecmqdfnt.MftNCyiY |
| Chain | Residue | Details |
| A | ALA96-TYR155 |






