7LA9
Crystal structure of the first bromodomain (BD1) of human BRD4 (BRD4-1) in complex with bivalent inhibitor NC-III-49-1
Functional Information from PROSITE/UniProt
site_id | PS00633 |
Number of Residues | 60 |
Details | BROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY |
Chain | Residue | Details |
A | ALA80-TYR139 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 6 |
Details | SITE: Acetylated histone binding => ECO:0000269|PubMed:22464331 |
Chain | Residue | Details |
A | ASN140 | |
B | ASN140 | |
C | ASN140 | |
D | ASN140 | |
E | ASN140 | |
F | ASN140 |
site_id | SWS_FT_FI2 |
Number of Residues | 12 |
Details | CROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733 |
Chain | Residue | Details |
A | LYS99 | |
F | LYS99 | |
B | LYS99 | |
C | LYS99 | |
D | LYS99 | |
E | LYS99 |