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7K7O

CRYSTAL STRUCTURE OF TYROSINE KINASE 2 JH2 (PSEUDO KINASE DOMAIN) COMPLEXED WITH COMPOUND-12 AKA:6-[(cyclopropanecarbonyl)amino]-4-{[2-methoxy-3-(pyrimidin-2-yl)phenyl]amino}-N-methylpyridazine-3-carboxamide

Functional Information from GO Data
ChainGOidnamespacecontents
A0004672molecular_functionprotein kinase activity
A0005524molecular_functionATP binding
A0006468biological_processprotein phosphorylation
B0004672molecular_functionprotein kinase activity
B0005524molecular_functionATP binding
B0006468biological_processprotein phosphorylation
Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for residue VZJ A 901
ChainResidue
AGLN597
AVAL690
AGLU691
AHIS692
AGLY693
AARG738
AASN739
ALEU741
ASER758
AGLY598
AVAL603
AVAL640
ALYS642
AALA671
ATHR687
AGLU688
ATYR689

site_idAC2
Number of Residues17
Detailsbinding site for residue VZJ B 901
ChainResidue
BLEU595
BGLN597
BGLY598
BVAL640
BLYS642
BTHR687
BGLU688
BTYR689
BVAL690
BGLU691
BHIS692
BGLY693
BARG738
BASN739
BLEU741
BSER758
BHOH1008

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Phosphotyrosine => ECO:0000250|UniProtKB:Q9R117
ChainResidueDetails
ATYR604
BTYR604

221716

PDB entries from 2024-06-26

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