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7K6R

Crystal structure of the bromodomain (BD) of human Bromodomain and PHD finger-containing Transcription Factor (BPTF) bound to GSK4027

Functional Information from GO Data
ChainGOidnamespacecontents
A0006357biological_processregulation of transcription by RNA polymerase II
A0016589cellular_componentNURF complex
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue 9ST A 3101
ChainResidue
ALEU2925
AHOH3247
APRO2951
APHE2952
APRO2955
AASP2960
ATYR3006
AASN3007
APHE3013
AHOH3210

site_idAC2
Number of Residues6
Detailsbinding site for residue EDO A 3102
ChainResidue
AVAL2967
ALYS2969
ATYR3005
AHOH3230
AHOH3276
AHOH3282

site_idAC3
Number of Residues3
Detailsbinding site for residue EDO A 3103
ChainResidue
AMET2922
ATHR2926
ATRP2950

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFlepvDpndap..DYYgvIkepMdlatMeervqrry..Yekltefvadmtk.IfdNCryY
ChainResidueDetails
AALA2949-TYR3006

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PDB entries from 2024-09-11

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