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7K0D

Crystal structure of the tandem bromodomain (BD1, BD2) of human TAF1 bound to mTORC1/2 inhibitor AZD3147

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0005669cellular_componenttranscription factor TFIID complex
A0006366biological_processtranscription by RNA polymerase II
A0016251molecular_functionRNA polymerase II general transcription initiation factor activity
A0017025molecular_functionTBP-class protein binding
Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue VQS A 1701
ChainResidue
APHE1405
AVAL1532
AASN1533
AVAL1537
ATYR1540
AASN1583
AVAL1413
ATYR1417
ASER1456
AASN1460
ATRP1526
APRO1527
AHIS1530
APRO1531

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues58
DetailsBROMODOMAIN_1 Bromodomain signature. TypFhtpvNakvvk..DYYkiItrpMdlqtLrenvrkrl..Ypsreefrehlel.IvkNSatY
ChainResidueDetails
ATHR1402-TYR1459
ASER1525-TYR1582

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PDB entries from 2024-06-12

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