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7FEE

Crystal structure of the allosteric modulator ZCZ011 binding to CP55940-bound cannabinoid receptor 1

Functional Information from GO Data
ChainGOidnamespacecontents
A0004930molecular_functionG protein-coupled receptor activity
A0004949molecular_functioncannabinoid receptor activity
A0007186biological_processG protein-coupled receptor signaling pathway
A0016020cellular_componentmembrane
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues25
DetailsTransmembrane: {"description":"Helical; Name=1","evidences":[{"source":"PubMed","id":"27768894","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27851727","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues30
DetailsTopological domain: {"description":"Cytoplasmic","evidences":[{"source":"PubMed","id":"27768894","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27851727","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues20
DetailsTransmembrane: {"description":"Helical; Name=2","evidences":[{"source":"PubMed","id":"27768894","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27851727","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI4
Number of Residues39
DetailsTopological domain: {"description":"Extracellular","evidences":[{"source":"PubMed","id":"27768894","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27851727","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI5
Number of Residues24
DetailsTransmembrane: {"description":"Helical; Name=3","evidences":[{"source":"PubMed","id":"27768894","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27851727","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI6
Number of Residues22
DetailsTransmembrane: {"description":"Helical; Name=4","evidences":[{"source":"PubMed","id":"27768894","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27851727","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI7
Number of Residues25
DetailsTransmembrane: {"description":"Helical; Name=5","evidences":[{"source":"PubMed","id":"27768894","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27851727","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI8
Number of Residues20
DetailsTransmembrane: {"description":"Helical; Name=6","evidences":[{"source":"PubMed","id":"27768894","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27851727","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI9
Number of Residues21
DetailsTransmembrane: {"description":"Helical; Name=7","evidences":[{"source":"PubMed","id":"27768894","evidenceCode":"ECO:0000269"},{"source":"PubMed","id":"27851727","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

243531

PDB entries from 2025-10-22

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