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7F8H

Structure-activity relationship studies of allosteric inhibitors of EYA2 tyrosine phosphatase

Functional Information from GO Data
ChainGOidnamespacecontents
A0004725molecular_functionprotein tyrosine phosphatase activity
A0007275biological_processmulticellular organism development
B0004725molecular_functionprotein tyrosine phosphatase activity
B0007275biological_processmulticellular organism development
C0004725molecular_functionprotein tyrosine phosphatase activity
C0007275biological_processmulticellular organism development
Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsActive site: {"description":"Nucleophile","evidences":[{"source":"PubMed","id":"19858093","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues3
DetailsActive site: {"description":"Proton donor","evidences":[{"source":"PubMed","id":"19858093","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues9
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"19351884","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

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PDB entries from 2025-08-13

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