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7C2Z

Bromodomain-containing 4 BD1 in complex with 3',4',7,8-Tetrahydroxyflavone

Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue SQH A 201
ChainResidue
APRO40
AVAL45
ALYS49
ALEU50
AASN98
AHOH327
AHOH339
AHOH373

site_idAC2
Number of Residues5
Detailsbinding site for residue FMT A 202
ChainResidue
AGLN20
AASN79
AALA80
AHOH378
ATHR18

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA38-TYR97

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues106
DetailsDomain: {"description":"Bromo 1","evidences":[{"source":"PROSITE-ProRule","id":"PRU00035","evidenceCode":"ECO:0000255"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues1
DetailsSite: {"description":"Acetylated histone binding","evidences":[{"source":"PubMed","id":"22464331","evidenceCode":"ECO:0000269"}]}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues2
DetailsCross-link: {"description":"Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2)","evidences":[{"source":"PubMed","id":"28112733","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

238895

PDB entries from 2025-07-16

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