Loading
PDBj
MenuPDBj@FacebookPDBj@TwitterPDBj@YouTubewwPDB FoundationwwPDB
RCSB PDBPDBeBMRBAdv. SearchSearch help

7B9O

Crystal structure of Retinoic Acid Receptor alpha (RXRA) in complexed with S169 inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0003707molecular_functionnuclear steroid receptor activity
A0005634cellular_componentnucleus
A0006355biological_processregulation of DNA-templated transcription
A0008270molecular_functionzinc ion binding
Functional Information from PDB Data
site_idAC1
Number of Residues19
Detailsbinding site for residue T72 A 501
ChainResidue
AILE268
ALEU326
AALA327
AILE345
APHE346
AVAL349
ACYS432
AHIS435
ALEU436
APHE439
AHOH601
AALA271
AGLN275
ATRP305
AASN306
AILE310
APHE313
AARG316
AILE324

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163, ECO:0007744|PubMed:24275569
ChainResidueDetails
AALA327
CTYR19

site_idSWS_FT_FI2
Number of Residues1
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:24275569
ChainResidueDetails
ASER259

site_idSWS_FT_FI3
Number of Residues1
DetailsMOD_RES: Phosphoserine; by MAPK8 and MAPK9 => ECO:0000250|UniProtKB:P28700
ChainResidueDetails
ASER260

221051

PDB entries from 2024-06-12

PDB statisticsPDBj update infoContact PDBjnumon