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7AXJ

Crystal structure of the hPXR-LBD in complex with estradiol and clotrimazole

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues8
Detailsbinding site for residue CL6 A 501
ChainResidue
ALEU209
AMET243
ASER247
APHE281
AGLN285
APHE288
ATRP299
AMET323

site_idAC2
Number of Residues7
Detailsbinding site for residue EST A 502
ChainResidue
ALEU206
ASER247
APHE251
AHIS407
AARG410
ALEU411
AASP205

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsBINDING: BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
ChainResidueDetails
AHIS407
ASER247
AGLN285

219869

PDB entries from 2024-05-15

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