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7AK1

Human MALT1(329-729) in complex with a chromane urea containing inhibitor

Functional Information from GO Data
ChainGOidnamespacecontents
A0004197molecular_functioncysteine-type endopeptidase activity
A0006508biological_processproteolysis
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue RJH A 801
ChainResidue
AVAL344
APHE398
ALEU401
AALA583
AGLN676
ALEU715
AMET717
AALA345
ALYS379
AVAL381
ALEU383
AGLU390
AASN393
AALA394
AGLU397

site_idAC2
Number of Residues5
Detailsbinding site for residue MG A 802
ChainResidue
AARG392
ACYS439
ALEU440
ACYS441
AASN444

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsACT_SITE: ACT_SITE => ECO:0000250
ChainResidueDetails
AHIS415
ACYS464

site_idSWS_FT_FI2
Number of Residues1
DetailsSITE: Breakpoint for translocation to form BIRC2-MALT1
ChainResidueDetails
AASP329

221051

PDB entries from 2024-06-12

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