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6ZC6

Small-molecule inhibitors of the PDZ domain of Dishevelled proteins interrupt Wnt signalling

Functional Information from GO Data
ChainGOidnamespacecontents
A0016055biological_processWnt signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue QEN A 401
ChainResidue
APHE259
AEDO404
ALEU260
AGLY261
AILE262
AVAL316
AARG320
AVAL323
AHIS324
AQEN402

site_idAC2
Number of Residues13
Detailsbinding site for residue QEN A 402
ChainResidue
ATYR257
AASN258
APHE259
APHE259
AGLY261
AMET282
AMET282
AGLY284
AGLY284
AGLY285
AQEN401
AEDO403
AHOH533

site_idAC3
Number of Residues2
Detailsbinding site for residue EDO A 403
ChainResidue
AQEN402
AHOH507

site_idAC4
Number of Residues3
Detailsbinding site for residue EDO A 404
ChainResidue
AASN258
AILE262
AQEN401

site_idAC5
Number of Residues4
Detailsbinding site for residue EDO A 405
ChainResidue
AVAL265
AILE278
AGLY296
AHOH521

238895

PDB entries from 2025-07-16

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