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6ZC4

Small-molecule inhibitors of the PDZ domain of Dishevelled proteins interrupt Wnt signalling

Functional Information from GO Data
ChainGOidnamespacecontents
A0016055biological_processWnt signaling pathway
B0016055biological_processWnt signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues15
Detailsbinding site for residue QEZ A 401
ChainResidue
AASN258
AVAL318
ALEU319
AARG320
AGLU321
AVAL323
AHOH533
APHE259
ALEU260
AGLY261
AILE262
AILE264
AASP314
AVAL316
AARG317

site_idAC2
Number of Residues10
Detailsbinding site for residue QEZ B 401
ChainResidue
AGLY266
ATYR277
BPHE259
BLEU260
BGLY261
BILE262
BVAL316
BARG320
BVAL323
BHOH513

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Symmetric dimethylarginine; by PRMT7; alternate => ECO:0000269|PubMed:23150776
ChainResidueDetails
AARG271
BARG271

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PDB entries from 2024-06-12

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