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6ZC3

Small-molecule inhibitors of the PDZ domain of Dishevelled proteins interrupt Wnt signalling

Functional Information from GO Data
ChainGOidnamespacecontents
A0016055biological_processWnt signaling pathway
B0016055biological_processWnt signaling pathway
Functional Information from PDB Data
site_idAC1
Number of Residues6
Detailsbinding site for residue EDO A 401
ChainResidue
AMET254
AGLU255
ALYS283
APRO326
AGLY327
AHOH507

site_idAC2
Number of Residues9
Detailsbinding site for residue JOR A 402
ChainResidue
AILE262
ALEU319
AARG320
AVAL323
AHIS324
AHOH535
APHE259
ALEU260
AGLY261

site_idAC3
Number of Residues11
Detailsbinding site for residue JOR B 401
ChainResidue
AGLU304
BPHE259
BLEU260
BGLY261
BILE262
BVAL316
BLEU319
BARG320
BVAL323
BHIS324
BHOH545

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsMOD_RES: Symmetric dimethylarginine; by PRMT7; alternate => ECO:0000269|PubMed:23150776
ChainResidueDetails
AARG271
BARG271

223790

PDB entries from 2024-08-14

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