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6YIL

Crystal structure of the CREBBP bromodomain in complex with a tetrahydroquinoxaline ligand

Functional Information from GO Data
ChainGOidnamespacecontents
A0004402molecular_functionhistone acetyltransferase activity
A0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues10
Detailsbinding site for residue OSQ A 1201
ChainResidue
APRO1110
AHOH1430
AVAL1115
ALEU1120
AASN1168
AARG1173
AVAL1174
AHOH1304
AHOH1364
AHOH1390

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. SlpFrqpvDpqllgipDYFdiVknpMdlstIkrkldtgq..Yqepwqyvddvwl.MfnNAwlY
ChainResidueDetails
ASER1108-TYR1167

223532

PDB entries from 2024-08-07

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