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6XUZ

CRYSTAL STRUCTURE OF BRD4-BD1 WITH COMPOUND 4

Functional Information from PDB Data
site_idAC1
Number of Residues14
Detailsbinding site for residue O1W A 201
ChainResidue
AARG58
AILE146
AHOH307
AHOH393
AHOH404
AHOH512
AGLN59
ATRP81
APRO82
APHE83
ALYS91
ALEU92
AASN117
AASN140

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140

site_idSWS_FT_FI2
Number of Residues2
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99

222415

PDB entries from 2024-07-10

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