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6XP9

STRUCTURE OF HUMAN PREGNANE X RECEPTOR LIGAND BINDING DOMAIN BOUND TETHERED WITH SRC co-activator peptide IN COMPLEX WITH (S,S)-1

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue QCG A 501
ChainResidue
AVAL211
ALEU239
AMET243
AMET246
AGLN285
APHE288
ATYR306
AMET323
AHOH657

site_idAC2
Number of Residues7
Detailsbinding site for residue GOL B 501
ChainResidue
AARG387
BTHR290
BLYS331
BLEU335
BHIS336
BGLU337
BHOH618

site_idAC3
Number of Residues10
Detailsbinding site for residue QCG B 502
ChainResidue
BVAL211
BLEU213
BLEU239
BMET243
BMET246
BGLN285
BPHE288
BTRP299
BTYR306
BHOH621

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues10
DetailsBinding site: {"evidences":[{"source":"PubMed","id":"12578355","evidenceCode":"ECO:0000269"},{"source":"PDB","id":"1M13","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

site_idSWS_FT_FI2
Number of Residues8
DetailsMotif: {"description":"LXXLL motif 4"}
ChainResidueDetails

site_idSWS_FT_FI3
Number of Residues1
DetailsModified residue: {"description":"Phosphoserine","evidences":[{"source":"PubMed","id":"23186163","evidenceCode":"ECO:0007744"}]}
ChainResidueDetails

245011

PDB entries from 2025-11-19

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