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6XP9

STRUCTURE OF HUMAN PREGNANE X RECEPTOR LIGAND BINDING DOMAIN BOUND TETHERED WITH SRC co-activator peptide IN COMPLEX WITH (S,S)-1

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006355biological_processregulation of DNA-templated transcription
B0003677molecular_functionDNA binding
B0004879molecular_functionnuclear receptor activity
B0006355biological_processregulation of DNA-templated transcription
Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue QCG A 501
ChainResidue
AVAL211
ALEU239
AMET243
AMET246
AGLN285
APHE288
ATYR306
AMET323
AHOH657

site_idAC2
Number of Residues7
Detailsbinding site for residue GOL B 501
ChainResidue
AARG387
BTHR290
BLYS331
BLEU335
BHIS336
BGLU337
BHOH618

site_idAC3
Number of Residues10
Detailsbinding site for residue QCG B 502
ChainResidue
BVAL211
BLEU213
BLEU239
BMET243
BMET246
BGLN285
BPHE288
BTRP299
BTYR306
BHOH621

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues6
DetailsBINDING: BINDING => ECO:0000269|PubMed:12578355, ECO:0007744|PDB:1M13
ChainResidueDetails
ASER247
AGLN285
AHIS407
BSER247
BGLN285
BHIS407

site_idSWS_FT_FI2
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0007744|PubMed:23186163
ChainResidueDetails
ASER461
BSER461

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PDB entries from 2024-10-09

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