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6X7D

BRD4 Bromodomain 1 in complex with multi-action inhibitor SF2523P

Functional Information from PDB Data
site_idAC1
Number of Residues9
Detailsbinding site for residue UT4 A 201
ChainResidue
ATRP81
APRO82
AGLN85
AVAL87
ALEU92
ALEU94
AASN140
AILE146
AHOH318

site_idAC2
Number of Residues5
Detailsbinding site for residue UT4 B 201
ChainResidue
BPRO82
BGLN85
BLEU94
BASN140
BHOH301

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140
BASN140

site_idSWS_FT_FI2
Number of Residues4
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99
BLYS99

224931

PDB entries from 2024-09-11

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