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6WE3

Human PARP14 (ARTD8), catalytic fragment in complex with compound 3

Functional Information from GO Data
ChainGOidnamespacecontents
A0003950molecular_functionNAD+-protein poly-ADP-ribosyltransferase activity
B0003950molecular_functionNAD+-protein poly-ADP-ribosyltransferase activity
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue TZ7 A 1901
ChainResidue
AHIS1682
ATYR1727
ALEU1782
AHOH2046
AGLY1683
AASP1685
ALYS1704
AALA1706
ATYR1714
ATYR1721
ASER1722
ATHR1726

site_idAC2
Number of Residues6
Detailsbinding site for residue EDO A 1902
ChainResidue
ATHR1631
ASER1634
ALYS1635
AGLN1638
APEG1908
ASO41913

site_idAC3
Number of Residues2
Detailsbinding site for residue EDO A 1903
ChainResidue
AHOH2069
AHOH2070

site_idAC4
Number of Residues3
Detailsbinding site for residue EDO A 1904
ChainResidue
ACYS1618
APRO1654
AHOH2001

site_idAC5
Number of Residues7
Detailsbinding site for residue EDO A 1905
ChainResidue
AVAL1689
AASN1693
AHOH2024
BPHE1617
BPRO1690
BASN1693
BHOH2023

site_idAC6
Number of Residues8
Detailsbinding site for residue EDO A 1906
ChainResidue
AASP1685
AALA1686
AGLY1687
AARG1729
ASO41912
ASO41912
AHOH2019
BEDO1904

site_idAC7
Number of Residues5
Detailsbinding site for residue EDO A 1907
ChainResidue
AASN1733
AARG1735
AHOH2035
BSER1700
BEDO1903

site_idAC8
Number of Residues6
Detailsbinding site for residue PEG A 1908
ChainResidue
AASN1630
ATHR1631
AEDO1902
AHOH2071
BSER1634
BASN1637

site_idAC9
Number of Residues2
Detailsbinding site for residue GOL A 1909
ChainResidue
ATRP1657
ATYR1792

site_idAD1
Number of Residues7
Detailsbinding site for residue GOL A 1910
ChainResidue
AGLY1696
APHE1697
ATYR1787
AASP1788
ATYR1789
AGLN1790
AALA1791

site_idAD2
Number of Residues3
Detailsbinding site for residue SO4 A 1911
ChainResidue
ALYS1678
AGLN1679
AHOH2005

site_idAD3
Number of Residues5
Detailsbinding site for residue SO4 A 1912
ChainResidue
AARG1729
AARG1729
AEDO1906
AEDO1906
BARG1729

site_idAD4
Number of Residues3
Detailsbinding site for residue SO4 A 1913
ChainResidue
ALYS1635
AGLN1638
AEDO1902

site_idAD5
Number of Residues12
Detailsbinding site for residue TZ7 B 1901
ChainResidue
BHIS1682
BGLY1683
BASP1685
BTYR1701
BLYS1704
BASN1705
BALA1706
BTYR1714
BTYR1721
BSER1722
BTYR1727
BLEU1782

site_idAD6
Number of Residues2
Detailsbinding site for residue EDO B 1902
ChainResidue
BLYS1635
BGLN1638

site_idAD7
Number of Residues6
Detailsbinding site for residue EDO B 1903
ChainResidue
AASN1733
AEDO1907
BHIS1691
BSER1700
BTYR1701
BLYS1704

site_idAD8
Number of Residues6
Detailsbinding site for residue EDO B 1904
ChainResidue
AASP1731
AALA1732
AEDO1906
BASP1685
BGLY1687
BARG1729

site_idAD9
Number of Residues5
Detailsbinding site for residue EDO B 1905
ChainResidue
BHOH2039
APRO1624
BPRO1624
BGLU1646
BHOH2005

site_idAE1
Number of Residues10
Detailsbinding site for residue PGE B 1906
ChainResidue
ALYS1647
AARG1735
AHIS1737
ATHR1798
BPRO1690
BHIS1691
BARG1694
BASN1695
BHOH2020
BHOH2023

site_idAE2
Number of Residues4
Detailsbinding site for residue PEG B 1907
ChainResidue
BGLN1652
BTRP1657
BTYR1792
BHOH2007

site_idAE3
Number of Residues5
Detailsbinding site for residue GOL B 1908
ChainResidue
BASN1616
BPHE1617
BCYS1618
BPRO1654
BHOH2022

site_idAE4
Number of Residues6
Detailsbinding site for residue GOL B 1909
ChainResidue
BLYS1664
BASP1668
BTHR1674
BMET1675
BASN1676
BGLU1677

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PDB entries from 2024-10-16

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