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6W9K

Structure of the Ancestral Glucocorticoid Receptor 2 ligand binding domain in complex with Prednisolone and PGC1a coregulator fragment

Functional Information from GO Data
ChainGOidnamespacecontents
A0003677molecular_functionDNA binding
A0004879molecular_functionnuclear receptor activity
A0006357biological_processregulation of transcription by RNA polymerase II
A0030518biological_processintracellular steroid hormone receptor signaling pathway
A0034056molecular_functionestrogen response element binding
Functional Information from PDB Data
site_idAC1
Number of Residues12
Detailsbinding site for residue TUA A 301
ChainResidue
ALEU32
ATHR208
AVAL216
APHE218
AASN33
AGLY36
AGLN39
AARG80
APHE92
AGLN111
APHE204
ACYS205

site_idAC2
Number of Residues5
Detailsbinding site for residue GOL A 302
ChainResidue
AGLU9
ASER76
AARG80
ATYR132
AHOH423

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues1
DetailsMOD_RES: N6-acetyllysine => ECO:0000250|UniProtKB:O70343
ChainResidueDetails
BLYS146

221051

PDB entries from 2024-06-12

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