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6VLH

HIV Integrase Core domain (IN) in complex with dimer-spanning ligand

Functional Information from GO Data
ChainGOidnamespacecontents
A0003676molecular_functionnucleic acid binding
A0015074biological_processDNA integration
B0003676molecular_functionnucleic acid binding
B0015074biological_processDNA integration
Functional Information from PDB Data
site_idAC1
Number of Residues2
Detailsbinding site for residue IOD A 301
ChainResidue
ALYS71
ALYS173

site_idAC2
Number of Residues2
Detailsbinding site for residue IOD A 302
ChainResidue
AHIS67
AGLY70

site_idAC3
Number of Residues2
Detailsbinding site for residue IOD A 303
ChainResidue
APHE121
AARG187

site_idAC4
Number of Residues3
Detailsbinding site for residue SO4 A 305
ChainResidue
ATHR66
AHIS67
ALYS159

site_idAC5
Number of Residues3
Detailsbinding site for residue SO4 A 306
ChainResidue
AASP116
AASN117
BGLU131

site_idAC6
Number of Residues4
Detailsbinding site for residue SO4 A 307
ChainResidue
ASER123
ATHR124
ATHR125
BLYS111

site_idAC7
Number of Residues6
Detailsbinding site for residue SO4 A 308
ChainResidue
APRO109
AHOH405
AHOH406
BTHR122
BLYS127
BLYS185

site_idAC8
Number of Residues1
Detailsbinding site for residue IOD B 301
ChainResidue
BLYS173

site_idAC9
Number of Residues3
Detailsbinding site for residue IOD B 302
ChainResidue
AARG199
AHOH421
BGLY70

site_idAD1
Number of Residues4
Detailsbinding site for residue SO4 B 303
ChainResidue
ATYR194
BTHR66
BHIS67
BLYS159

site_idAD2
Number of Residues4
Detailsbinding site for residue SO4 B 304
ChainResidue
BLYS159
BILE162
BGLY163
BARG166

site_idAD3
Number of Residues6
Detailsbinding site for residue SO4 B 305
ChainResidue
BSER57
BPRO58
BGLY59
BILE60
BLYS111
BHOH423

site_idAD4
Number of Residues4
Detailsbinding site for residue SO4 B 306
ChainResidue
BSER123
BTHR124
BTHR125
BHOH409

site_idAD5
Number of Residues3
Detailsbinding site for residue SO4 B 307
ChainResidue
BILE60
BGLN62
BHIS114

site_idAD6
Number of Residues23
Detailsbinding site for residue R2A B 308
ChainResidue
AGLU87
AGLN95
AGLU96
AALA98
ATHR125
AALA128
AALA129
AALA169
AGLU170
AHIS171
ALYS173
ATHR174
AMET178
BGLN95
BGLU96
BTYR99
BLEU102
BTHR125
BALA129
BALA169
BGLU170
BHIS171
BTHR174

219869

PDB entries from 2024-05-15

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