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6VIW

BRD4_Bromodomain1 complex with pyrrolopyridone compound 18

Functional Information from PDB Data
site_idAC1
Number of Residues16
Detailsbinding site for residue QYV A 201
ChainResidue
ATRP81
ALEU94
ATYR139
AASN140
AILE146
AHOH304
BTRP81
BQYV201
APRO82
APHE83
AGLN85
APRO86
AVAL87
AASP88
ALYS91
ALEU92

site_idAC2
Number of Residues15
Detailsbinding site for residue QYV B 201
ChainResidue
ATRP81
AQYV201
BTRP81
BPRO82
BPHE83
BGLN85
BVAL87
BLEU92
BLEU94
BASN140
BASP145
BILE146
BMET149
BHOH301
BHOH307

site_idAC3
Number of Residues13
Detailsbinding site for residue QYV C 201
ChainResidue
CTRP81
CTRP81
CPRO82
CPHE83
CGLN85
CPRO86
CVAL87
CASP88
CLYS91
CLEU92
CASN140
CILE146
CHOH302

Functional Information from PROSITE/UniProt
site_idPS00633
Number of Residues60
DetailsBROMODOMAIN_1 Bromodomain signature. AwpFqqpvDavklnlpDYYkiIktpMdmgtIkkrlenny..Ywnaqeciqdfnt.MftNCyiY
ChainResidueDetails
AALA80-TYR139

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues3
DetailsSITE: Acetylated histone binding => ECO:0000269|PubMed:22464331
ChainResidueDetails
AASN140
BASN140
CASN140

site_idSWS_FT_FI2
Number of Residues6
DetailsCROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733
ChainResidueDetails
ALYS99
BLYS99
CLYS99

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PDB entries from 2024-10-16

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