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6V2S

Crystal Structure of chromodomain of MPP8 in complex with inhibitor UNC3866

Functional Information from PDB Data
site_idAC1
Number of Residues17
Detailsbinding site for UNC3866 chain C
ChainResidue
AVAL58
AHOH321
BMET67
BLYS68
BTHR69
BARG107
BALA111
CHOH101
CHOH102
APHE59
AGLU60
AVAL61
ATRP80
ATYR83
AGLU91
AHIS95
AGLU101

site_idAC2
Number of Residues16
Detailsbinding site for UNC3866 chain D
ChainResidue
ALEU104
AARG107
ALYS108
BASP57
BVAL58
BPHE59
BGLU60
BVAL61
BTRP80
BTYR83
BASP87
BGLU91
BHIS95
BASP98
BCYS99
BHOH310

Functional Information from PROSITE/UniProt
site_idPS00598
Number of Residues21
DetailsCHROMO_1 Chromo domain signature. YkVRWkGYtsddd.TWEPeihL
ChainResidueDetails
ATYR76-LEU96

Functional Information from SwissProt/UniProt
site_idSWS_FT_FI1
Number of Residues2
DetailsSITE: Interaction with histone H3K9me3 => ECO:0000269|PubMed:21419134
ChainResidueDetails
APHE59
BPHE59

site_idSWS_FT_FI2
Number of Residues2
DetailsMOD_RES: Phosphoserine => ECO:0000250|UniProtKB:Q3TYA6
ChainResidueDetails
ASER85
BSER85

218853

PDB entries from 2024-04-24

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