6V1E
Crystal structure of the bromodomain of human BRD7 bound to BI7273
Functional Information from PDB Data
site_id | AC1 |
Number of Residues | 12 |
Details | binding site for residue 5SW A 301 |
Chain | Residue |
A | SER153 |
A | ASN211 |
A | TYR217 |
A | HOH413 |
A | ALA154 |
A | PHE155 |
A | PHE156 |
A | PHE158 |
A | PRO159 |
A | VAL160 |
A | PHE163 |
A | ILE164 |
site_id | AC2 |
Number of Residues | 7 |
Details | binding site for residue EDO A 302 |
Chain | Residue |
A | ILE171 |
A | ILE172 |
A | LYS173 |
A | HIS174 |
A | LEU202 |
A | ASN206 |
A | GLU235 |
Functional Information from SwissProt/UniProt
site_id | SWS_FT_FI1 |
Number of Residues | 6 |
Details | CROSSLNK: Glycyl lysine isopeptide (Lys-Gly) (interchain with G-Cter in SUMO2) => ECO:0007744|PubMed:28112733 |
Chain | Residue | Details |
A | LYS186 | |
A | LYS197 | |
A | LYS201 | |
A | LYS212 | |
A | LYS241 |